ZempiloAmalungiselelo

"Risperidone": imiyalelo ukusetyenziswa. "Risperidone Organic": inkcazelo, izimvo, Izimo

Age, utshintsho zengqondo kunye yokuziphatha kunokuba nzima kakhulu ubomi kuphela umntu ogulayo, kodwa isangqa wangaphakathi. Unyango lwezifo psychogenic kunye nezinye yinkqubo engelula, kodwa iyeza le nto, yimani ngxishi, ceba ephakadeni iindlela ezintsha ukujongana nawo. Eyona ndima ephambili unikwa unyango. Tablets "Risperidone" analogs leyo baninzi kakhulu, aphakathi iimveliso kakhulu zithandwa. Yintoni phawu wabo? Indlela ukuthatha kubo, yaye ukuba unayo nayiphi na Izimo? Ngaba ndisebenzisa ezi pilisi nokudakumba? Iimpendulo zale mibuzo siza kuzama ukunika kweli nqaku.

ifomu Release komsindo "Risperidone" iziyobisi

"Risperidone" Amacwecwe enziwe kwakhona ziinkampani ezininzi zamachiza phantsi kwegama elifanayo yaye kakhulu ukwakhiwa efanayo. Eyona nto iphambili ebonakalayo ichiza okunene ngokwayo risperidone xa isixa-1, 2 okanye 4 mg (ngokuxhomekeke balawule). tablet nganye isale inwebu ama-camera emhlophe. tablet ngeenxa zonke, biconvex. In cross-candelo ibonisa ngokucacileyo maleko ezimbini: i nomphandle wocango. Ukubunjwa amacwecwe "Risperidone" - ukongeza esisebenza - kuquka amacandelo ezongezelelweyo: starch, lesilicon dioxide, nemagnesium stearate kunye MCC.

Tablets "Risperidone" kunye analogs zabo, kuquka "Organics Risperidone", eyenziwe iiphakheji Inkcazo iziqwenga 10 nganye, nayo, zingafakwa kwiibhokisi zekhadibhodi Imiqulu-2, 3, 5 okanye 6 kunye imiyalelo ukuze isicelo. imveliso Ukudibanisa obuvelisiweyo kunye sibuphethe ngezitya kwiglasi emnyama, ngalinye ezo ziquka amacwecwe-20, 30, 50 okanye 60. Iibhanki nawo zingafakwa kwiibhokisi ikhadibhodi ne myalelo.

wenza njani imithi?

I yangoku umyalelo 'Risperidone "iipilisi into ebhekiselele bensizoksazola, okt neuroleptics. Ukongeza isiphumo antipsychotic eli chiza, sine hypothermic kunye neempawu antiemetic. Oku kungenxa kukukwazi ukuvala isithako esebenzayo D2-zemizwa Mesocortical kunye neenkqubo mesolimbic kunye neziko emetic, kwaye kananjalo kuchaphazela receptors adrenergic eyendayo esikhondweni ebuchotsheni. Kwakhona umchiza uyakwazi ukuvala receptors dopamine kule ngxenye.

Ngenxa propati amayeza le "Risperidone" amanqaku lweziyobisi phantse lonke HIV, unako ukucinezela iimpawu ukuphazamiseka neurogenic ezifana iimfeketho zokufeketha kunye nemibono, ndlongondlongo kunye ukuzenzekela. Phantsi kwale mvelaphi, iingcali qaphela ukuba chiza phantse akukho alunasiphumo kwi umsebenzi iimoto, kodwa ngaxeshanye, ofihla iimpawu kwangumqondiso Uthando ngesifo sengqondo.

Distribution kunye kukhuthaza

Le nokwenziwa osisiqu esebenzayo kwisiqwenga zesisu lwenzeka ngexesha elifutshane kwaye inani. ekudleni na inkqubo vliyaetetot. Ubuninzi agxile kwi plasma yegazi arhente esebenzayo ifikelela neyure emva ezithatha ichiza. Ahlobene njengoko risperidone (-hydroxyrisperidone 9) bathi bafakwe ngokucothayo.

Ngokuphathelele ukusasazwa beziyobisi emzimbeni "Risperidone" yemiyalezo ithi malunga kwii ukwimo esebenzayo zomzimba ezahlukeneyo kunye namalungu, kwaye ingqondo, kunye nobisi lwebele. Unxibelelwano kunye iiproteni plasma kule meko malunga ne-90%.

Half-ubomi beziyobisi Kwenzeka ngezigaba ezimbini: ngethuba leeyure ezi-3 kufuphi-70% ye-compound idubule yi izintso ekwimo ingaguqukanga, lo gama i-digidrorisperidon 9 ukuboniswa phantse imini yonke. izigulane abadala kunye nabo abaphethwe ukusilela kwezintso, nexesha kukhuthaza beziyobisi landa.

Sebenzisa beziyobisi: zikhombisa kunye Izimo

Faka ichiza "Risperidone" umyalelo manual icebisa ukuba xa zifo zilandelayo okanye ukuphazamiseka emzimbeni:

  1. uhlobo Acute okanye engapheliyo ngesifo sengqondo.
  2. disorder Psychopathic, luphawulwa obubonakala kakubi okanye elinemveliso nomqondiso.
  3. Izigulo zempilo yengqondo, kunye kweepesente ezingama.
  4. IDementia ngokuqhelekileyo ebangela uqhambuko ngumsindo ndlongo, iimfeketho zokufeketha kunye nezinye iimpawu ngengqondo.

Kwakhona ziboniswa abantwana elivisayo babo babe nendawo disorder (utyekelo etshabalalisayo) ukukhubazeka izangoma okanye engqondweni, ngokunjalo enokuphazamisa disorder mania lwaya neziyobisi "Risperidone". Kule meko, eli cwecwe lidlala indima exhasayo kulo unyango.

Oko ikhona kwi Izimo neziyobisi ezibalulekileyo eziquka hypersensitivity ukuba amacandelo amacwecwe. Ukongeza, ichiza "Risperidone" yemiyalezo ucebisa ukusebenzisa ngononophelo kakhulu kwi izifo okanye miqathango ilandelayo:

  • yamathumba ingqondo kunye ithombo legazi yobuchopho;
  • ukusilela hepatic kunye kwezintso kwifomu kakhulu;
  • ukuphazamiseka patency isisu;
  • isifo sentliziyo, kuquka iposi engabalulekanga, ukusilela intliziyo, ezingapheliyo block ifomu antrioventikulyarnaya kunye bradycardia;
  • Drug libanda, okanye ukuxhomekeka phezu kwabo;
  • emzimbeni;
  • isifo Parkinson kaThixo;
  • uphathwe (ngexesha ichiza okanye isifo);
  • Ukukhulelwa ne zisanyisa.

Ngaphaya koko, eli chiza ayikhuthazwa "Risperidone" (amacwecwe) zokudakumba, nto leyo ichazwe kwi ukuncitshiswa umsebenzi nomonde bafune ukuzibulala. Kwakhona nabantu ngenyameko prescribers yakhe yobudala sele ayifikelelekanga kwiminyaka eli-15.

Umthamo kunye nendlela owamkeleka

Oyidlayo kunye neendlela ixhomekeka ichiza iyafumaneka kwi sisifo yesigulane, ubungqongqo ukuvuza, kwaye kukho izifo ezihamba okanye States zophendlo lwezifo. Zonke iinkcukacha ezifanelekileyo malunga nokusetyenziswa "Risperidone" iziyobisi ungabona le theyibhile.

Isifo okanye imeko

balawule

Notes isicelo

schizophrenia

ithamo Ukuqalisa - 1 mg 2 amaxesha ngemini. Ithamo kwi we2 Kwiintsuku ezilandelayo ngu 4 mg (2 umphinda mg 2 ngosuku).

Ukuba i "Risperidone" ichiza wamiselwa indawo namanye amachiza, akulula xa uqeqeshelwa ukuba kufuneka kwenziwe kancinci.

Esiyingozi sengqondo kunye nezinye naresheniya ubudala

1 mg ngosuku, ukuba ichiza kufuneka 1 ixesha ngosuku.

Phambi ukuphazamiseka kwendlela umsebenzi wezintso kwaye ithamo wesibindi kuncitshiswa ngu 2 umphinda-, ngokwenyusa kancinane de kucetyiswa.

Mania, kwengqondo okanye ezinye ukuphazamiseka kwengqondo

Ukuqala yedosi - 2 mg ngosuku (ngenye imini yokwamkela), ngoko ithamo ebegqwese Linyuke ku-6 mg ngosuku.

Nceda uqaphele le lekhefu phakathi nokunyuka ithamo ntsuku ezi-2.

izifo lezimilo olufikisayo

1 mg ngosuku, ukwamkelwa olulodwa

ubunzima yesigulane kufuneka bungabi ngaphantsi kwe-50 kg, kwimeko malungana idosi kufuneka alungiswe.

ukukhubazeka engqondweni ngasemva ukuphazamiseka kwengqondo etshabalalisayo

1 mg ngosuku

Xa ingozi ebalulekileyo mania kunye nokunciphisa efunekayo gipermany ithamo yokuqala ukunyuka okuthe chu ukuya Kunconywa.

mayingagqithi 16 mg nasiphi na isifo okanye imeko ukulungiselela ngemihla ithamo "Risperidone".

abasabela Ezingalunganga kumzimba kunye libanda

Enye into ebalulekileyo ukuba kufuneka wazi izigulane bajamelene ikhondo unyango with "Risperidone" - side effects esinokubakho kule nkqubo yokwamkela iipilisi. Amathuba kwazo kuxhomekeke ikakhulu phezu ngamnye. Ngoko ke, yintoni kumphazamisa umguli?

Amaninzi kuvela abasabela ilandelayo evela amalungu kunye neenkqubo ezahlukeneyo:

  • usulelo lwe iphecana eliphezulu bokuphefumla wokuchama (ingakumbi izigulane abadala unesifo "iDementia");
  • intloko, ukuphazamiseka kwendlela ubuthongo, isiyezi, ukozela kunye ukungaboni;
  • ukuqunjelwa, iintlungu epigastric, isicaphucaphu, umlomo owomileyo;
  • ukuphazamiseka Intliziyo rhythm (tachycardia);
  • nokudumba le isifo ngeempumlo kunye ityhubhu Eustachian, apho isigulane uziva impumlo ukuvaleka okanye iindlebe, impumlo kuchitheka igazi;
  • ukukhohlela, impumlo esihambisayo, kwakunye nokubamba-bamba umphefumlo;
  • igazi;
  • ngumchamo womchamo;
  • ukudumba kwamalunga, utshintsho iqinelwa (ingakumbi kubantu abalupheleyo), iqolo ubuhlungu.

kukho kwakhona iqela ziziphumo ebezingalindelekanga, ezo kuthelekiswa kunqabile kwenzeka "Risperidone" ezithatha ichiza. Iingcali Ukubuyekezwa bathi phakathi kwabo kulandelayo:

  • indlebe kunye neso izifo;
  • amagciwane echaphazela umzimba wonke okanye endawo;
  • womchamo yokuphefumla, kuquka inyumoniya, tonsils, iphika kunye tracheobronchitis;
  • onychomycosis kunye acrodermatitis;
  • ukudideka, ixhala, mania kunye hypomania, zeDyskinesia;
  • izihlunu nokoma, nokushisa, ukwanda ukubila;
  • oscillations ezingazinzanga wegazi;
  • sokuwa;
  • belele, umgudu eliphezulu occlusion isikhohlela (neempempe ngexesha yokuphefumla, rales zimanzi okanye dysphonia);
  • ukwandisa okanye ukunciphisa ubunzima;
  • Izitenxo sexesheni, ukungabikho ukuchama, priapism, ukungabi namdla ngokwesondo;
  • bomzimba ebeleni izihlunu;
  • ukudumba kwesikhumba, ingakumbi ubuso, kuthibaza, unxano, chaza influenza-ezifana;
  • ubuthathaka iingalo kunye nemilenze, nokuziva ukuqina kwamalunga.

Kwimeko yendlela kakhulu emibi ezithatha ichiza "Risperidone" ntonye beziyobisi akufunekanga ibe indawo ufanele ukuba amayeza, njengoko ziqulathe izithako ezifanayo ezisebenzayo. Kulo mzekelo, i ingcali kuya ukhethe kwelinye ichiza, nto leyo ubunjwe kusitsha, okanye amayeza ezongezelelweyo ukuze kupheliswe neempawu ezingemnandi.

Iimpawu kunye nonyango lwe libanda, iziyobisi

Xa imiyalelo ezingafanelekanga iidosi ukuya phezulu libanda Inokwenzeka, nto ichazwa ngendlela lwaziwayo gqolo ukwehlisa uxinzelelo lwegazi kunye neengxaki zentliziyo isingqisho (tachycardia). Ukongeza, isiguli uphazamise somnolence, ukulalisa, iingxaki ezinxulumene nokuphefumla kunye disorder extrapyramidal.

iyeza ngqo ekulungiseleleni "Risperidone" hayi, ngoko unyango lujoliswe ngokususa mpawu kakhulu libizwe. Njengoko uncedo kwisigulana yokuqala kufuneka ihlanjwe esiswini kwaye wamalahle isebenza kunye laxatives. Ngokunciphisa uxinzelelo lwegazi imithetho ezibalulekileyo ifuna ulawulo efakwa of agonists kunye nezisombululo nokubandakanywa.

Kulo lonke ixesha elifunekayo esweni kwentliziyo ukuba ukubona iintlobo ezahlukeneyo arrhythmias inhliziyo. Ukuba naliphi na elibhaqiweyo, uthomalaliso amayeza afanelekileyo.

imiyalelo engqalileyo ngokusebenzisa ichiza

Xa ekufumaneni ichiza "Risperidone" yemiyalezo ucebisa ukuba balandele isikhokelo ezimbalwa ezibalulekileyo. Oku akuyi kuphela kunciphisa amathuba neziphumo ebezingalindelekanga, kodwa ukuphucula imeko yeli isigulana phambi co-morbidities.

Kuqala ufuna ukunikela ingqalelo ngokukhethekileyo umthamo ichiza kwabo izigulane kuye kukho izifo kwinkqubo sentliziyo. Kulo mzekelo, ichiza ekuqaleni lolwamkelo eyimfuneko iingedosi ezincinane, ngokuthe ngcembe zakhuliswa ukuba amaxabiso ezinqwenelekayo. Iziphakamiso efanayo kwimeko hypovolemia, emzimbeni kunye nezigulo cerebrovascular.

Iingcali kwakhona ukuba luyeke ukusetyenziswa nokudla-calorie ukudla hlobo. Oku kubangelwa kukuba unyango lwe "risperidone" iziyobisi amathuba aphezulu iseti ubunzima engaphezulu.

Ayikhuthazwa ngexesha iipilisi unyango "Risperidone 'ukuba benze imisebenzi enxulumene nolawulo izithuthi kunye nezinye iindlela ezifuna yoxinaniso yomguli eziphakamileyo kunye reactions lengqondo ngokukhawuleza.

Intsebenziswano kunye namanye amachiza

Xa kutyunjwa ichiza "Risperidone", ixabiso apho kuya kuxoxwa kamva, kufuneka athathe ingqalelo ubuchule layo ukusebenzisana ngamayeza amaninzi. Kwezinye iimeko, oku kunokukhokelela iziphumo ezingalindelekanga kwaye mnandi kakhulu. Ngenxa yoko, iziyobisi, xi ukusebenza luvo abantu, ngokunjalo ethanol, kunye ne "Risperidone" bamqumbise ukwimeko enjalo, njengoko isongezo CNS imisebenzi kukudakumba.

Amanye amachiza, ezifana beta-blocker, abaninzi, zonke, ngaphandle kokukhetha, lakhula tricyclic nga kwandisa ukufumaneka ukwimo "Risperidone" amacwecwe esebenzayo kwi plasma yegazi. Kunjalo kweyeza "Fluoxetine". "Carbamazepine", phezu koko, kunciphisa uyondelelwano lwee- into esebenzayo lithetha "Risperidone" plasma. Xa ukuqeshwa kwabo joint kufuna esweni rhoqo isigulane, kwakunye nokunciphisa kwirejimeni nomthamo.

reviews

Izimvo amacwecwe "Risperidone Organics" yaye "Risperidone", ixabiso leyo kuthathwa ukuba zibe nokufikeleleka kubantu kuluhlu olubanzi abathengi (umlinganiselo engange 170 pack nganye), azikwazi kubizwa ngokuba negative. Isiphumo ukuba amacwecwe izifo ezahlukeneyo psychogenic okanye indlela yokuziphatha, umbono ezintle zombini iingcali kunye nezigulane. aphendule nje kunye analogs kweli chiza, ngenxa yokuba kwiimeko ezininzi umahluko phakathi kwe zimbini kuphela sixa-mali kunye nokwakhiwa phantse efanayo (ngaphandle excipients).

Amacwecwe ethile ebalulekileyo kuphela "Risperidone" (analogs ngezixhobo esebenzayo nabo bawe phantsi le nkcazelo) - ezininzi ziziphumo ebezingalindelekanga, leyo kwezinye iimeko ezinokuchaphazela umgangatho yomguli ngayo ubomi ngcono. Yiyo loo nto iingcali bacebisa xa elivela kuzo naziphi abasabela emibi qhagamshelana nogqirha wakho ukuze wabelane naye ukufumana indlela yokuphuma kule meko.

Ngoko, sifunde ukuba ziphi iipilisi "i-Risperidon". Umyalelo, intengo, izifaniso kunye nokuphendula kakubi kwezinto eziphilayo zaqwalaselwa ngokucacileyo kweli nqaku. Ekugqibeleni, ndingathanda ukukhumbula ukuba le nkunkuma isasazwa kuphela kwi-odokotela. Ukulawulwa okungagunyazisiweyo nokulawulwa kwamacwecwe eli qela kunokulimaza impilo yakho.

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