Zempilo, Amalungiselelo
Naiz (ekhompyutheni) - yemiyalezo.
ifomu balawule
Amalungiselelo yenziwa ngeendlela drug-3 - ukumiswa, amacwecwe esasazekayo kunye eqhelekileyo. Ukunqunyanyiswa yi ivumba elithozamisayo okunomnyinyivane mthubi ngebala kunye kakhulu uphawu ukungcamla kweli chiza. Ukunqunyanyiswa unako redispersed xa beshukumisa igutyana.
Iipilisi zenziwa phantse emhlophe, kunye namona kancinane elityheli. Amacwecwe ngokwemilo setyhula, biconcave, imiphezulu zayo zombini smooth.
UDenise ukwakheka:
ukumiswa
into esebenzayo
- Nimesulide - 50 mg (5 ml yokumisa)
Excipients:
- sorbitol
- glucose
- gum xanthan
- propyl
- methylparaben
- citric acid
- yi isongo
- WS umbala Yellow
- glycerol
- polysorbate
- ngamanzi okuhlamba
amacwecwe esasazekayo
into esebenzayo
- Nimesulide - 50 mg (Itheyibhile 1).
excipients
- aspartame
- calcium phosphate
- microcrystalline kwincindi
- carboxymethyl starch
- corn starch
- talc
- wemagniziyam stearate
- Colloidal electronic dioxide
- yi isongo
tablets
into esebenzayo
- Nimesulide - 100 mg (Itheyibhile 1).
Excipients:
- wemagniziyam stearate
- Calcium Hydrogen Phosphate
- microcrystalline kwincindi
- electronic Anhydrous colloidal
- corn starch
- Sodium starch glycolate
- talc lihlanjululwe
Isenzo amayeza ye ichiza
inyathelo amayeza ubalisa kuqala UDenise - iipilisi, lo myalelo iqulethe iinkcukacha kokwamkelwa kwazo zonke iifom balawule. Ichiza eli NSAID, equlethe kwayo amaqela isakhiwo sulfonilidnuyu. kungenzeka Nimesulide kunxulumene inhibitors of Cox-2, ukuze lineziphumo anti-ezithintela ukosuleleka kunye iintlungu, ukongeza, ichiza usebenzisa iziphumo iintlungu, kodwa isidanga engaphantsi.
Indlela yokusebenza ye ichiza ezinxulumene kwezithandani le Yindibanisela prostaglandins e nokudumba kwezithandani ye ukuyilwa radicals ioksijini kunye inhibition yokukhululwa myeloperoxidase.
Pharmacokinetics
UDenise sathatha ngokugqibeleleyo ukusuka iphecana zesisu, ufikelela iphezulu egazini sele emva iiyure ezi-2. Ichiza yi 99% ziiprotein ebembophile.
Ukulungiselela babantu - tablets isikhokelo iyathathwa kwimithombo ezisemthethweni, metabiliziruetsya esibindini kwaye kwazona kwi umchamo, nge 98% ye idosi unikwe imveliso emini.
ubungqina
- izifo rheumatism ephuhlisa ngaphandle philisi joint
- ukudleka
- Nangokurhala, njalo emva kotyando
- Pain okubangelwa seTrojan
- Fever kunye ubuhlungu xa ukudumba etsolo kwi yomoya eliphezulu
imiphumela Side UDenise
Tablets, umyalelo apho ngoku, unako ukuvelisa icala elingenzi nto- kwiinkqubo ezahlukeneyo kunye namaziko:
iziphumo ebezingalindelekanga ichiza, ezinxulumene lokugaya
- isizothe-zothe
- heartburn
- nesisu esibuhlungu
- ilindle ungalibali
iziphumo ebezingalindelekanga ichiza, ezinxulumene inkqubo luvo:
- ikhanda
- ukozela
- nesiyezi
iziphumo ebezingalindelekanga ichiza, ezinxulumene negazi lakho:
- erythema
- ufunga
- urticaria
Eminye imiphumela emibi:
- Ukugcinwa kwi incindi yomzimba
- oliguria
- ayanda
Izimo UDenise
Ngaba uluhlu Izimo kucetyiswa apho ukuphepha ezithatha ichiza, yaye xa kuyimfuneko, kuphela emva kokudibana nogqirha wakho.
- Ukopha evela iphecana zesisu
- ukusilela kwezintso
- ukusilela hepatic
- Ukukhulelwa ne zisanyisa
- isifo Peptic zesisu
Drug ukwenzelana babantu
Tablets, imiyalelo malunga nokusetyenziswa awo ntoni kukhokelela data epheleleyo kwaye olubanzi yonke imithi kuqulunqo ngolu hlobo lulandelayo: hayi kucetyiswa ne-arhente zilandelayo - phenytoin, digoxin, naziphi womchamo, iziyobisi lithium, anticoagulants, iziyobisi umfutho, NSAIDs, methotrexate, cyclosporin .
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