Zempilo, Amalungiselelo
Ichiza "stugeron" yesikhokelo.
Ichiza "stugeron": Ifom release, isakhiwo nokupaka
Amacwecwe ezimhlophe, iflethi, ngeenxa zonke, kunye esisodwa, ukuba phantse akukho ivumba, kwicala elinye - othi "STUGERON", amashumi amabini anesihlanu neemiligram isithako esebenzayo - cinnarizine, namadyungudyungu emacwecweni amabini anesihlanu mahlanu. Ukubunjwa ibandakanya, ukongeza cinnarizine, kwaye okunye: dust colloidal, iitapile starch, nemagnesium stearate, talc, povidone, umbona starch, monohydrate lactose.
Imiphumo amayeza beziyobisi "stugeron" yemiyalezo ikuchaza ngale ndlela ilandelayo.
Oku kunciphisa ukungena ion calcium kwizisele, ithowuni Imisonto kwezihlunu kwamagingxi sisezindongeni arterioles, iphucula isiphumo Ukuthanjiswa iinqanawa carbon dioxide kunye nangaphezulu. Ngenxa ichiza "stugeron" iimpembelelo ngqo kwi nemithambo egudileyo izihlunu, ukuba uyakwazi ukwehlisa abasabela ngayo zizondlo (epinephrine, angiotensin, dopamine, vasopressin). It has a isiphumo vasodilating (ingakumbi ngokuphathelele iimpahla Cerebral), kodwa ube nefuthe elibi kwixabiso uxinzelelo lwegazi. umsebenzi Imiboniso antihistaminic luchaphazela inkqubo vestibular, ukuhla excitability yayo, kunye nenkqubo onovelwano luvo, lisibekele ilizwi layo. Kwakhona kubangela ukwanda luthambe erythrocyte inwebu kunye nokukwazi kwabo ukugqabhuza, ekunciphiseni viscosity igazi. Ukongeza, izihlunu umzimba kwandisa kwinkcaso hypoxia.
Le pharmacokinetics beziyobisi "stugeron" umyalelo zokusetyenziswa uchaza kunjalo.
Resorption beziyobisi lwenzeka kwi emathunjini kunye nesisu. Le xi okungaphezulu e plasma emva kulawulo ichiza ngaphakathi kufikelelwa ngokusebenzisa esinye - Iiyure ezintathu. iiproteni plasma okubopha alithoba ananye ekhulwini cinnarizine. Metoboliziruet ukulungiselela (by glyukuronirovaniya) ngokupheleleyo esibindini. ixesha bawo-ubomi iiyure ezine. Metabolites tsinnarizina output wesinye kwisithathu yi nezintso, kwaye isibini-yethumbu.
Le umthamo ncwadana "stugeron" umyalelo kweziyobisi unika oku kulandelayo.
Thatha kufuneka abe, emva kwesidlo. Xa ukuphazamiseka ebuchotsheni kwegazi - ezingamashumi amabini anesihlanu - milligrams amahlanu (omnye - amacwecwe amabini) izihlandlo ezithathu ngosuku. Xa izifo yegazi peripheral - mahlanu - milligrams asixhenxe anesihlanu (ezimbini - iipilisi ezintathu) izihlandlo ezithathu ngosuku. Kwaye kwimeko ukuphazamiseka vestibular - ezingamashumi amabini anesihlanu milligrams (elinye icwecwe) izihlandlo ezithathu ngosuku. Xa "indlela" kwesi sifo (kinetoses) - esithathwa abadala - ezingamashumi amabini anesihlanu milligrams, isiqingatha seyure phambi kokuba uhambo (ukuba kuyimfuneko, kusafuneka ukuba ukuthatha iiyure njengoko ezintandathu), "stugeron" abantwana kwiimeko ezinjalo, anike malunga nesiqingatha ithamo ekucetyiswa abantu abadala. Kwimeko apho hypersensitivity ukuya kwenye amacandelo ichiza "stugeron" yemiyalezo ekucetyiswa ukuba ukuqala unyango kunye isiqingatha idosi, ngokuthe ngcembe zandise oko. Ikhosi konyango ngokuqhelekileyo ithatha iiveki ukuya kwiinyanga. Elona nani liphezulu sivumelekile ngemihla manual idosi "stugeron" umyalelo unika milligrams ezingamakhulu amahlanu okanye tablets ezisithoba.
Kwimeko libanda - isisu wabandezeleka uhlanjiweyo acocekileyo amanzi, nika namalahle yasebenza.
Ukuba ichiza emiselweyo "stugeron 'abantwana?
Ukuphonononga kumsebenzi womnatha zinxulumene ikakhulu ukuqeshwa kwakhe Encephalopathy osana evela hypoxia ezingekazalwa, kwakunye kwi the CNS sisilonda esidumbileyoesingaphakathi osana kunye syndrome of neuro-reflex excitability. Uphawula indlela ethile emihle. Kuchaziwe ngugqirha kumnika ikota elucwecweni kabini ngemini emva kokutya, grinded xa ngecephe kunye nomxube ukondla okanye ekupheleni lokondla. Ekupheleni - nika yentsalela eselwayo Umxube okanye emanzini.
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