ZempiloAmalungiselelo

Ichiza "Terfenadine": imiyalelo yokusebenzisa

Yeyiphi kufuna isixhobo ezifana 'Terfenadine "? Imiyalelo yokusebenzisa, ixabiso, ncomo, kunye nolawulo konwaywa ichiza zidweliswe ngezantsi. Ukongeza, eli nqaku linika ulwazi malunga iimpawu ichiza wathi, analogue zayo Izimo.

ifomu Release kunye namacandelo kuthetha amacandelo

Ziziphi ifomu yenziwe amayeza "Terfenadine"? Imiyalelo lithi isicelo ukuba ichiza ifumaneka azipilisi, leyo eziqulathe isithako esebenzayo ezifana terfenadine. Ukongeza, i-arhente isifundo akhululwayo ngokohlobo ukunqunyanyiswa yolawulo yomlomo, isiraphu kunye nomgubo crystalline ilungiselelwe isisombululo.

iimpawu imithi

Yintoni eyanceda "Terfenadine"? Imiyalelo Sebenzisa ithi le antihistamine. Kubalulekile ukwazi ukuba zivale ngokukhetha engabalulekanga receptors H1-histamine nokuthintela ukwandiswa emithanjeni nokwandisa permeability zabo, aqaqambayo agudileyo, kuquka bronchoconstriction kubantu nesi sifo, uphuhliso erythema, angioedema kunye ukurhawuzelela.

Isiphumo emva kokufaka olu nyango kubonakala emva kweeyure ezimbini yaye ifikelela incopho yayo emva ezine. Noko ke, waligcina ezinesiqingatha ngosuku.

Xa nokuthimliswa uyalisa iziyobisi esebenzayo lula kwaye kucutha nezihlandlo nokuthimla, yaye kunciphisa ukurhawuzelela, rhinorrhea kunye epiphora.

Ezinye iimpawu ichiza

Yintoni ephawulekayo na indlela ngokuthi "Terfenadine"? Imiyalelo yokusebenzisa (amayeza ixabiso eliboniswe ngezantsi) uthi ukuba eli chiza ukusebenza anticholinergic eliphakathi kunye iibhloko imiphantsi (potassium) cardiomyocytes kwaye attenuates ubukhali bronchospasm.

A ukwanda okubonakalayo egazini terfenadine usenokuphelekwa ukwandiswa kwexesha QT kunye nophuhliso iziganeko ezinkulu inhliziyo.

ikhono kinetic

Njengoko ichiza ako ngokukhawuleza "Terfenadine"? Imiyalelo phezu ithi isicelo ukuba oku kuthetha ifunxwe ukusuka phecana zesisu ngokukhawuleza. Oku kumiselwa i-plasma yegazi emva kwemizuzu engama-30.

Eli chiza enebana iiproteni plasma yi-97%. It awulungelelananga ezetyiswa ngayo sisibindi kunye nokusekwa metabolites ezimbini.

Medicine "Terfenadine" isebenza ngokufanayo kuwo onke amaqela izigulane, kungakhathaliseki ubudala babo.

ubungqina

Kwezinye iimeko, ukumisela amayeza "Terfenadine"? Imiyalelo yokusebenzisa kweengxelo ukuba indlela ephumelelayo kakhulu nokuthimliswa ngamaxesha kukwalisa, conjunctivitis negazi, urticaria ezondeleyo idiopathic, nangokhwekhwe atopic, qhagamshelana dermatitis, irhashalala kunye ukurhawuzelela okubangelwa isifo sesibindi. Kwakhona medicament esebenzayo ezimiselweyo angioedema, negazi zibangelwa ngamayeza, ziinyosi isinambuzane kunye nokutya, isifuba kunye umkhuhlane (kuphela kwanonyango zidityaniswe).

Ukongeza, eli chiza isoloko isetyenziswa xa ukuthintelwa nokwaliwa, babonakaliswa xa kubhalwa eendaba umahluko.

Uvala ukuqashwa

Medicine "Terfenadine" contraindicated ukuba ayayamkela hypersensitivity, hypokalemia, hypomagnesemia, kululwa interval QT kwi-ECG, zolwaphulo ezivakaliswa esibindini kwaye abantwana (ukuba azipilisi - iminyaka emithandathu, yaye oluludaka - ukuya kwiminyaka emithathu).

Drug "Terfenadine": imiyalelo yokusebenzisa

Analogs of medicament zidweliswe ngezantsi.

Uthe kuthetha wamisa abadala ingaphakathi abantwana ukusuka kwiminyaka mg elinambini ukuya kuma-60 kabini yonke imihla okanye 120 mg kanye ngemini. Inani inkulu ichiza efunyenweyo iiyure eziyi-24 ngu-480 mg.

Abantwana iminyaka 6-12 yi iyeza emiselweyo mg 30 kabini ngemini, kunye namatakane eminyaka 3-5 imisiwe kukho umthamo 15 mg kabini ngemini.

Iintshukumo ngu-lomsebenzi

Ukulungiselela unyango i "Terfenadine" izigulane zinokuba iziganeko ezingalunganga ezifana:

  • ubuthathaka, iyangongoza, intloko ebuhlungu, kululwa QT lekhefu, isiyezi;
  • tachyarrhythmia ventricular, ukuphazamiseka ekulaleni, arrythmia, ukozela, fibrillation ventricular, uvalo;
  • ukudakumba, zokuma, ifiva, hypotension, hematopoiesis kakuhle, niphele;
  • thrombocytopenia, unditsho, kome na isifo somlomo, paresthesia, kwanda, ukungaboni, ukuqunjelwa;
  • bronchospasm, isicaphucaphu, inwebu eyomileyo kwiinwebu le empumlweni nasemqaleni, ukugabha, khohlo, ukungakhululeki esiswini, umqala obuhlungu;

  • kutshintsha kwi-frequency isitulo, nokopha, cholestasis, rhoqo ukuchama, nenyongo, seTrojan, hepatitis;
  • lafa, irhashalala, urticaria, nangokhwekhwe, photosensitivity, iinwele ukuxozwa, angioedema, alopecia;
  • galactorrhea, anaphylaxis, ukubila.

Analogue, ixabiso, ncomo

analogue Drug kuthathwa "uhambo" yaye "Bronal". Price of ichiza malunga 190-215 engange nganye amacwecwe-10.

Nohlolo "Terfenadine" ukulungiselela ubukhulu becala HIV. Izigulane babanga ukuba kuthetha kakuhle ukumelana ezahlukeneyo negazi lakho. Bobubi kweli chiza ziquka ubukho neziphumo zakhe ebezingalindelekanga.

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