ZempiloAmalungiselelo

Yintoni "ibuprofen" (tablets)? "Ibuprofen" - ijeli, amafutha, ukunqunyanyiswa: yesikhokelo, ncomo. "Ibuprofen" (isiraphu abantwana): imiyalelo yokusetyenziswa

Yintoni "ibuprofen" emiselweyo kwizigulana? Oku kuya kukuxelela kwinqaku langoku. Kuwo uya kufunda indlela athi yenziwe ngaluphi na uhlobo, idosi kufuneka athathwe njalo njani kwaye yintoni.

Ubume, ukupakishwa, inkcazelo, iintlobo ichiza

wavelisa "ibuprofen" Ngayiphi indlela? Imiyalelo yokusebenzisa, iingcali yokwenene ingxelo ukuba eli chiza lukhutshwe ngeendlela ezahlukeneyo.

  • Amacwecwe ngeenxa Biconvex kwaye ziyafumaneka ukuthengiswa iibhokisi-20, 10 okanye amaqhekeza 100. Bathi umgangatho ogudileyo namhlophe. Le into esebenzayo yale ichiza ibuprofen.
  • Camera "ibuprofen" iipilisi. Ukususela oko ezi pilisi, siza kukuxelela phambili umganyana. Ziqulethe uluhlu imali encinane element esebenzayo, ngaloo ndlela kubonelelwa inyathelo ngokuzinzileyo.
  • Njengezingxobo. Le fom iqulethe mg 300 of into esebenzayo. Baya ukunyibilika ngokucothayo kakhulu.
  • "Ibuprofen" nokumiswa. Isiraphu abantwana lufumaneka ezithengiswayo kwibhotile ngecephe yokulinganisa. Ukunqunyanyiswa yi ubunzima yohlobo olunye lwe umbala omthubi. Kusenokuba, njengoko isongo-orenji nestrawberry.
  • "Ibuprofen" suppositories. Imiyalelo, ukubuyekeza bathi ezi amakhandlela zisetyenziswa rectally. Bona kuthengiswa iipakethe iziqwenga ezili-10.
  • Zithutha. Le fomu lokulungiselela kwesisombululo medicament ngenxa yokufakwa. Le mveliso ogqityiweyo uba incasa minty kunye livumba elithozamisayo.
  • "Ibuprofen" 5%, linamafutha aqholiweyo. Ukusetyenziswa kwale sixhobo sikuvumela ukuba kukuphelisa uqaqanjelwa imisipha namalungu. Le gel lisetyenziswa ngokwemixholo kuphela.
  • A isisombululo ngenaliti. It yenziwa eJamani babethengisa imiqulu ngekhadibhodi njengezingxobo 4. Faka iziyobisi yegazi.

Iimpawu beziyobisi

Yintoni "ibuprofen" lisetyenziswa yezonyango? Ngokutsho imiyalelo, ichiza a nonsteroidal arhente anti-ukudumba. Uyakwazi ukuba ekuphembeleleni i anti-ukudumba, antipyretic kunye neziphumo iintlungu. Iingcali zithi le sixhobo njee iibhloko TSOG2 kunye TSOG1.

Umgaqo inyathelo ibuprofen kuyehla prostaglandin yokuqaphela, oko kukuthi, njengabalamli nangokurhala, iintlungu kunye nempendulo hyperthermic.

Pharmacokinetics beziyobisi

Zeziphi pharmacokinetic iparameters ziye "ibuprofen" tablet? Iifom zesicelo se kuqulunqo ngomlomo iqinisekisa ukufakwa eliphezulu kwaye ukuzila ukusuka phecana zesisu.

Ukufumaneka eliphezulu ibuprofen kwi plasma emsebenzini emva kwemizuzu 120-240 emva nolawulo. Unxibelelwano protein plasma ngaphezu kwama-90% kunye nesiqingatha ubomi - 2 hr.

Drug "ibuprofen" (ukunqunyanyiswa kunye tablets) kancinci lingena singene amalungu. impahla yawo asebenzayo bazondelele kule inyama synovia. Oku kunika kube nokuqwalaselwa eziphakamileyo esisebenza.

Emva ukufakwa malunga ne-60% ye engasebenziyo R-uhlobo ichiza similise okwaloo esebenzayo S-imilo.

Eli chiza umzimba. Isiphumo ngayo nge izintso (singaguqukanga), yaye kunye enyongweni.

Iimpawu zibonisa ukuba ukusetyenziswa kwaso nasiphi na isiyobisi

Yintoni "ibuprofen" elinokunikwa izigulane? Ngokutsho imiyalelo, eli chiza Yayibubungqina zilandelayo:

  • Ukuphazamiseka spinal, kunye nezigulo yokukrala amalungu (kubandakanywa ankylosing spondylitis, isifo samathambo kunye sifo, osteoarthritis);
  • syndrome febrile, ezenzeka imvelaphi yazo njengomkhuhlane ezosulelayo okanye;
  • intlungu ngokulinganisela imvelaphi ezahlukeneyo (kuquka intloko ebuhlungu, neuralgia, migraine, iintlungu postoperative, iintlungu wamazinyo, myalgia, isifo sephepha zaseprayimari, iintlungu post-traumatic).

"Ibuprofen" unokusetyenziswa nawuphi na umyalelo kodwa? Ukususela oko ezi pilisi lalathelwe ukuba izigulane? Oogqirha bathi oku ichiza ngokubonakalayo eyayisetyenziselwa impilo nomqondiso. Yena kakuhle yaye ngokukhawuleza kunciphisa nokudumba kunye neentlungu (kuphela ngexesha lokusetyenziswa), kodwa aluchaphazeli ukuqhubela phambili kwesifo.

Izimo

Yintoni "ibuprofen" iyasetyenziswa, izigulane, siye ezichazwe apha ngasentla. Ngokuphathelele Izimo, ngoko ke ziquka umguli kulandelayo:

  • ilunga nezifo sisilonda ye phecana wokudla, ingakumbi kwisigaba etsolo (umz, isilonda-12 tiperstnoj emathunjini, isisu, isifo Crohn kaThixo, sisilonda sikabhobhosi, nonspecific);
  • hypersensitivity yabantu izithako ezenza ichiza;
  • hypersensitivity ogulayo acetylsalicylic acid kunye nezinye NSAIDs, kuquka imbali yezonyango nokuthimliswa, fit inyumoniya, urticaria emva NSAID okanye acetylsalicylic acid;
  • isifo wamathumbu arhabaxa;
  • buso okanye epheleleyo acetylsalicylic acid ukunganyamezelani syndrome (wabonakalaliswa njengoko rhinosinusitis, urticaria, polyp kwi isifo ngeempumlo, isifuba inyumoniya);
  • ixesha emva kwemithambo esa igazi;
  • sophele diathesis, kubazali kunye nezinye izifo ekunqandeni egazini (umzekelo, hypocoagulation);
  • ukusilela kakhulu hepatic, izifo ezahlukeneyo esibindini;
  • yokopha intracranial, ukopha zesisu;
  • severe insufficiency kwezintso, ukuqinisekisile hyperkalemia;
  • isifo esiqhubekayo sezintso.

Ziziphi ezinye Izimo zikhona "ibuprofen 'iziyobisi? Isiraphu abantwana ayikhuthazwa ukunika iintsana phantsi iinyanga ezi-3, kunye nezinye iintlobo amayeza - kwiminyaka emi-6. Kwakhona, le iyeza kufuneka ingasetyenziswa ngexesha lokukhulelwa.

wamkelekile ukuqapha

Kuphantsi kwaziphi iimeko apho kufuneka emiselweyo amayeza "ibuprofen" ngononophelo obukhulu? Application (feedback ngale sixhobo iza kwenziwa kamva) beziyobisi abadala, kunye nabantu abane sisifo sentliziyo, umfutho wegazi kunye nesifo sentliziyo kobuchopho kufuneka bagadwe ngeliso elibukhali ngugqirha wakho.

Kwakhona ngononophelo obukhulu banikwa amayeza ezimiselweyo isifo cerebrovascular, dyslipidemia, isifo seswekile, izifo kwemithambo (peripheral), ukutshaya, enteritis, ukuselwa kotywala rhoqo, ukuqina kwesibindi, gastritis, nephrotic syndrome, hyperbilirubinemia, ukudumba, izifo egazini imvelaphi ongaziwayo nasebudeni webele ibele.

Iindlela isicelo beziyobisi

Iindlela Ukusetyenziswa ichiza ixhomekeke kwiifomu yayo ukukhululwa.

  • Isiraphu.

Ziziphi oyidlayo iyaboniswa "ibuprofen 'abantwana? Imiyalelo Sebenzisa ithi, ngokunxulumene emacwecweni, isiraphu wenza kakhulu ngokukhawuleza. Ngaphambi ngokusebenzisa le fomu Shake kakuhle. Le umthamo ichiza kufuneka ichaze kuphela wezingane, ngokuxhomekeke imeko yesigulane.

  • Amakhandlela.

Suppositories "ibuprofen" eyenzelwe ngokukodwa iintsana. Zisetyenziswa rectally, aze aqalise ukwenza emva kwemizuzu engama-30. Xa fever okanye intlungu syndrome, idosi enye ye- ichiza 5-10 mg ngamnye 1 kg ubunzima umntwana. Sebenzisa ikhandlela ngokukhethekayo kudluliswe iiyure 6-8.

  • Gel, linamafutha aqholiweyo.

Ndingayisebenzisa njani le nkcitho yamafutha "ibuprofen"? Le gel strip 1.5 cm esisetyenziswe sisilonda esidumbileyoesingaphakathi massage mnene. Kuyinto umtsalane ukuphepha ukudibana nesiyobisi inwebu yangaphakathi kunye amanxeba avulekileyo. Kungenjalo, le medicament efunekayo nangoko pula ngamanzi ashushu.

  • Amacwecwe.

Ngaba "ibuprofen" iipilisi eziyingozi kubantwana? Imiyalelo Sebenzisa ithi olu hlobo ichiza akufuneki ukuba amatakane ukuya kwiminyaka emi-6.

Thatha olu nyango kufuneka ibe phakathi nokutya. Ngokuqhelekileyo, oko ibhalwa isixa 5-10 mg 1 kg ubunzima bomzimba nganye kathathu ngemini. Ngoko ke, lo idosi yemihla ngemihla ukuba ngaphezu kwama-20 mg kg nganye.

Xa isifo samathambo kunye nezinye izifo edibeneyo, ichiza elo lilawulwa isixa-40 mg / kg (kodwa hayi ngaphezulu).

amacala libanda

Xa amathamo aphezulu ichiza alandelayo iimpawu nazo kwizigulane: isicaphucaphu, silale, iintlungu esiswini, ukozela, ukugabha, ukuduma, ukudakumba, lactic metabolic, intloko ebuhlungu, ukusilela etsolo kwezintso, angabikho zingqondweni, bradycardia, sinciphise uxinzelelo lwegazi, fibrillation atrial imithambo, yima zokuphefumla tachycardia.

Unyango - lavage engxamisekileyo esiswini (kwimizuzu engama-60 emva kokuba libanda), ulawulo wamalahle luvuliwe, kwaye diuresis amanzi obrak.

imiphumela emibi

Ngaba ukubonakala ezibi reactions iziyobisi "ibuprofen"? Gel ukusetyenziswa lwangaphandle soze kubangela iziphumo ezingafunekiyo. Ngokumalunga iintlobo yomlomo ichiza, zinokubangela ezi ziphumo zilandelayo:

  • iintlungu esiswini, ukungabi namdla, isicaphucaphu, umlomo isibetho, ukugabha, gingival isifo zizilonda, pyrosis, stomatitis aphthous, urhudo, kome okanye kwinwebu emlonyeni, flatulence, pancreatitis, ukuqhina;
  • hepatitis;
  • bronchospasm, dyspnea
  • endlebeni, ingxolo okanye unkenteza ezindlebeni, ubuthulu;
  • ukuluma kwaye kome yamehlo, scotoma, izilonda yityhefu ye-luvo optic, ukungaboni kabini okanye ukungaboni, udumba iinkophe kunye conjunctiva;
  • sokulibala, intloko ebuhlungu, ukuba nemibono, isiyezi, ukudideka, ixhala, badandatheke, ukuba nochuku kunye uvalo, somnolence, ukuphazamiseka, aseptic meningitis;
  • tachycardia, ukusilela intliziyo congestive, uxinzelelo oluphezulu lwegazi;
  • ukusilela etsolo kwezintso, polyuria, nephritis negazi, nephrotic syndrome, Ngokuzimela;
  • irhashalala, angioedema, pruritus, erythema multiforme anaphylactoid reactions, ifiva, anaphylaxis, dyspnea, bronchospasm, Stevens-Johnson syndrome, eosinophilia, epidermal necrolysis ityhefu, nokuthimliswa umzimba;
  • ukwanda ukubila;
  • anaemia, purpura thrombocytopenic, kunye thrombocytopenia, leukopenia, agranulocytosis;
  • zizilonda ukopha zesisu.

Kufuneka kuqatshelwe ukuba yokwamkela yokulungiselela kunokubangela utshintsho amanani alandelayo laboratory:

  • serum creatinine xi (ukwanda);
  • ukopha ixesha (ukwanda);
  • ukucoca creatinine (kunciphisa);
  • xi glucose serum (ukuncipha);
  • athwala okanye hematocrit (ukuze lincitshiswe);
  • umsebenzi isibindi transaminase (ukwanda).

Xa isenzeko ngayo ezinjalo kufuneka ngoko nangoko ezithatha ichiza aze adibane nogqirha.

izincomo ezithile

amayeza Unyango "ibuprofen" kufuneka yenziwe idosi ubuncinane ukuba baya kubonisa ukusebenza eliphezulu nezinyangayo. Kule khosi unyango kufuneka ibe mfutshane.

Ukuba unyango lwenziwa ixesha elide, kuthatha kolawulo izintso wesibindi kunye nomfanekiso igazi peripheral.

Ukuba iimpawu gastropathy kufuna esweni ngenyameko imeko yesigulane. Kufuneka kubandakanya nokuqhutywa esophagogastroduodenoscopy, kwakunye ilindle uvavanyo lwegazi ubugqi kunye wegazi epheleleyo (ukumisela yetekisi).

imithi

Kuyinto ukulungiselela ehlangene ikhokela "ibuprofen" aspirin kwakunye nezinye NSAIDs. Oku kungenxa yokuba kunganciphisa iziphumo ukudumba kwaye antiplatelet kwezi arhente.

Ngelo xesha ezithatha ichiza wenzelwa le ngxelo iziyobisi thrombolytic kwaye anticoagulant kwandisa umngcipheko ukopha.

"Tsefaperazon", "Tsefamandol" valproic acid 'tsefotetan "yaye" plikamitsin "kwandisa amathuba okuba nesifo gipoprotrombinemii.

Iziyobisi ezithintela secretion tubular, ukunciphisa zinomgutyulo nokwandisa plasma yoxinaniso of "ibuprofen".

medicament kujongwa isidima isenzo arhente uricosuric, iphucula iimpembelelo anticoagulants, fibrinolytics kunye arhente antiplatelet.

Imithi Izigulane '

Drug "ibuprofen" into ethandwa kakhulu phakathi izigulane. endaweni yayo njenge arhente ngempumelelo kakhulu anti-ukudumba ukuba unalo iintlobo ezahlukeneyo woyekelelo.

Ngokutsho iimpendulo yezigulane, iyeza liqala ukwenza ngokukhawuleza kakhulu. Isusa nkqu intlungu kakhulu kakhulu kwamalungu kunye nemisipha, kwaye ishenxisa yintloko kunye ukudumba imvelaphi ezahlukeneyo.

Le ethile kuphela kule iyeza linani elikhulu yeziphumo ebezingalindelekanga kunye Izimo. Ngokutsho iimpendulo lezigulane, "ibuprofen" iziyobisi badla kunokubangela iintlungu esiswini, isicaphucaphu, isiyezi kunye nokugabha, kwaye uba unobangela izilonda kunye erosions kwi lokugaya. Ngoko ke, sebenzisa eli chiza xa ubuncinane umlinganiselo ekucetyiswa kunye ixesha elifutshane. Indlela kuphela uya kukwazi ukuphelisa intlungu yaye uvakalelwa naziphi na iziphumo ebezingalindelekanga.

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