ZempiloAmalungiselelo

Ichiza "Spitomin": imiyalelo ukusetyenziswa, izalathisi, Izimo

Namhlanje ke ndithi kuni ngalo eli chiza, njengoko "Spitomin". Imiyalelo yokusebenzisa, ixabiso, ncomo, analogs kunye neempawu zayo - zonke ezi zihlandlo zizigulane abanomdla ukuba ugqirha emiselweyo olu nyango. Lonke ulwazi oluyimfuneko inokufumaneka kamva kweli nqaku.

Inkcazelo ichiza, ukumila kwayo, kunye nokwakheka zizinto ebekupakishwe

Yintoni na ichiza "Spitomin"? Imiyalelo yokusebenzisa (ukulungiselela echazwe kukho thaca ngokweenkcukacha olukhulu) uthi le ipilisi esha emhlophe, imilo setyhula kwaye iflethi, kunye chamfer kunye Valium kunye nemiqadi «E151».

Isixhobo iqulethe hydrochloride buspirone kunye namacandelo abangabancedani ezifana wesitatshi carboxymethyl, monohydrate lactose, nemagnesium stearate, isodiyam, microcrystalline neselulosi kunye dust colloidal anhydrous.

Ekuthengisweni beziyobisi kuza Imiqulu blister kunye iibhokisana.

isimiso ukusebenza

Ziziphi iimpawu ezikhoyo iziyobisi "Spitomin 'na? Imiyalelo yokusebenzisa (amacwecwe ixabiso thaca ngezantsi) uthi ukuba le arhente anxiolytic, ebhekiselele kuthotho non-benzodiazepine kwaye isiphumo bucala.

Ngokungafaniyo nezinye anxiolytics, eli chiza na antiepileptic, sine thile kunye neempawu myorelaxant. Umgaqo yayo yokusebenza isekelwe phezu imiphumo buspirone kwi dopaminergic kunye serotonergic neenkqubo.

Oku kuthetha emane evalela i receptors dopamine (presynaptic) kwaye kwandisa izinga excitation zemithambo-luvo (dopamine) ephakathi.

Ziziphi ezinye iipropati ezendeleyo iziyobisi "Spitomin"? Imiyalelo yokusebenzisa ithi Buspirone i agonist uyakhetha kwenxenye ye-5-HT1A receptor serotonin. Oku akuchaphazeli nomphetho receptors benzodiazepine kunye Gaba, yaye akuyi kuchaphazela umsebenzi lengqondo akubangeli nokunyamezelana. Ukongeza, esi sixhobo asikusebenzeli potentiate ifuthe iziselo ezinxilisayo.

Isiphumo therapeutic beziyobisi ingqalelo phuhlisa ngcembe yaye kwenzeka emva omnye okanye emibini emva unyango.

Kinetics izimali

Kukufakwa ichiza "Spitomin", imiyalelo zokusetyenziswa oboniswe ngezantsi, kwenzeka kwisiqwenga zesisu. Buspirone awulungelelananga umzimba ngexesha nokuwela esibindini. bioavailability sayo-4% kwaye plasma yoxinaniso eliphezulu ekufikelelwe kuso emva kweyure enye.

Buspirone iyekelela kunye nobisi. Ukuze ufumane inkcazelo malunga kwii-ichiza ngokusebenzisa njengomqobo placental kusilela.

Ukulungiselela zivela ilindle iiyure ezintlanu.

ubungqina

Ukususela oko kumiselwe "Spitomin" tablet? Imiyalelo yokusebenzisa lubonisa okukhomba zilandelayo:

  • syndrome kwekhono yawo;
  • nexhala sifo jikelele;
  • ekubalekeni syndrome utywala (njengoko unyango adjuvant);
  • one- ;
  • izifo depressive (njengoko unyango adjuvant).

Izimo

Kwezinye iimeko, ayikhuthazwa tu into yokuba ukusebenzisa iipilisi 'Spitomin "? Imiyalelo yokusebenzisa uthi ezimbi zilandelayo nemiqathango phantsi apho ithamo iyeza contraindicated ku:

  • glaucoma;
  • hypersensitivity ukuba izithako ichiza;
  • myasthenia gravis;
  • insufficiency kwezintso, kakhulu;
  • yobudala minor;
  • ukwamkelwa ngaxeshanye Mao inhibitor ;
  • zisanyisa;
  • ngexesha lokukhulelwa.

Nge arhente care ibhalwa esibindini kwesibindi kunye ukusilela kwezintso.

Medicament "Spitomin": imiyalelo yokusebenzisa

Analogs beziyobisi uya thaca ngezantsi.

Of iimali ekufuneka athathwe ngexesha elifanayo ngosuku, phambi okanye emva kwesidlo.

Ichiza Akuvunyelwe ukusebenzisa athile (xa kukho imfuneko) ukuba unyango ixhala, kuba isiphumo yayo zonyango iphuhlise ukusetyenziswa kuphela emva ngokuphindaphindiweyo.

Esithathwa yale iyeza esikhethwe ngamnye. Ngokuqhelekileyo, akukho 15 mg. Kufuneka yahlulwe 2-3 nasebusuku.

Ithamo iphezulu enye i-30 mg kwaye ubuninzi ngemihla - 60 mg.

Xa abadala kufuneka i-hlengiso umthamo. Xa medicament kakuhle kwezintso okanye hepatic kufuneka isetyenziswe ngokuqaphela ngeedosi ezincinane.

imiphumela emibi

Ngokuqhelekileyo amayeza "Spitomin 'Wanyamezela kakuhle. Kuphela kwezinye iimeko, esi sixhobo na ukunyhashwa ezithile:

  • iintlungu esifubeni, yokulala, niphele, isiyezi, hypotension, intloko ebuhlungu, hypertension;
  • ixhala luvo, ukuphazamiseka ebuchotsheni yokujikeleza, reactions dysphoric, decompensation ukungaphumeleli kwentliziyo, ukwanda uvakalelo ingxolo, iposi engabalulekanga, ongase, cardiomyopathy, yokuzibulala, bradycardia;
  • depersonalization, ukunyamezelana ebandayo, imincili, bephelelwa, hyperkinesis, ukuduma, ixhala, ukurhawuzelela emehlweni, silale, iliso bomvu, nemibono, abanale, ukudideka, ukuphazamiseka ngengqondo;
  • ukungaboni, laryngitis, conjunctivitis, udumba isifo ngeempumlo, incasa kakuhle, imvakalelo ubunzima esifubeni, ukuphazamiseka indlebe engaphakathi, hyperventilation, iintlungu iliso, ukungabikho umoya, photophobia, epistaxis, ukwanda koxinzelelo intraocular;
  • galaktoreyu, isicaphucaphu, umonakalo lengqula, flatulence, enuresis ebusuku, ukudla, ukwanda wokutya, dysuria, ukuvuza izinkcwe, ukuphazamiseka sexesheni, ukopha isisu, ukuchama kwalibaziseka kunye nezinye.

Price, analogue, ncomo

Indleko yale arhente imalunga 600 engange. Ukuba kuyafuneka, nto ithathwa analog ezifana "Buspirone Sandoz."

ncomo Consumer yazisa ukuba ichiza uchaphazelekayo arhente elungileyo anxiolytic. Noko ke, oko kuthatha i ingcali kuphela injongo ixesha elide (hayi ngamaxesha athile).

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