Ichiza "Buserelin Long" i analogu zokwenziwa of hormone yendalo GnRH. Utyando esi sixhobo inokhuphiswano ngqo njengesibophelelo kwi receptors kwiiseli yebhinqa kunye ekwandeni ezidlula msinyane kumazinga steroid ngesondo kwi-plasma, nto leyo ekugqibeleni kukhokelela ukuvaleka olupheleleyo ekuthiwa gonadotropic umsebenzi yebhinqa. Ngenxa ichiza "Buserelin Long" ibonelelwa abathintela ngqo hormone kudibaniso kwi gonads, esizibonakalisa njengoko ukuhla kumanqanaba testosterone (indices post-kuthenwa) kumadoda nokunciphisa estradiol igazi post-ngxaki iimpawu kwizigulana ababhinqileyo. Kwimeko yokuqala sonke sithethe xa kuthenwa amayeza, elinesibini - on postmenopausal okanye ovariectomy.
Iyeza, uyakhululwa ngomzuzwana nje lyophilizate eyenzelwe ngokukodwa ukulungiselela oluludaka. Ukwakhiwa kwale ukulungiselela njengento engundoqo kuquka malunga 4 mg buserelin acetate. components Auxiliary sodium carmellose, a copolymer of glycolic kunye DL-lactic acid, polysorbate-80 kunye d-mannitol.
Ngokumalunga ukusetyenziswa kweziyobisi, i-arhente elimisiweyo "Buserelin Long 'ukuba unyango umhlaza webele kunye enama-oxhomekeke umhlaza wendlala. Ukongeza, eli chiza ingasetyenziswa ngexesha unyango lwe endometriosis. Kuba unyango lwe fibroids zesibeleko kunye ubudlolo (ngokusebenzisa inkqubo-IVF) Kwakhona kufuneka uqale ukusebenzisa iziyobisi "Buserelin-Long". Izimvo oogqirha engqinela iziphumo ezilungileyo ukusetyenziswa kwayo ukuze unyango kweenkqubo endometrial hyperplastic.
Ukuba sithethe malunga Izimo eziphambili ukusetyenziswa, ngoko sebenzisa olu nyango contraindicated ngqo kubantu ngabanye ukunganyamezelani buserelin acetate, kwakunye naziphi na ezinye iindawo kuyo axhasayo. Ukongeza, Izimo ziquka ukukhulelwa kunye zisanyisa.
Ngokwahlukeneyo, kufuneka athi malunga iziphumo ebezingalindelekanga kunokwenzeka zokusetyenziswa kwemali "Buserelin-Long", njengoko kunokuba, umzekelo, unobangela urticaria, nokudumba angioneurotic kunye hyperemia. Ukongeza, kusenokuba kukho iimeko ezifana demineralization, ukuphazamiseka kokulala, intloko ebuhlungu kunye nokudakumba. Xa izigulane ababhinqileyo iintlungu esiswini, utshintsho yobuntu, ukubila ukwanda, menstrualnopodobnye ukopha kwaye kome le isifo langasese ngenxa yokusebenzisa iziyobisi eyenziweyo "Buserelin-Long". side effects emadodeni zinxulunyaniswa ikakhulu kunye exacerbation kwezifo engundoqo, ukugcinwa wokuchama, gynecomastia, yaye "kidney ukudumba." Ukongezelela, oko kuphawulwa ukuncipha amandla, ukubila ukwanda, buthathaka kwezihlunu yesiqephu kunye ithambo iintlungu. A Inani elincinane izigulane ukusabela ezifana neengxaki zesisu , kunye Embolism nezengekho miphungeni.