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Ichiza "Betagestin" ukusuka vertigo. "Betahistine": imiyalelo ukusetyenziswa, ixabiso, ncomo

wenza ichiza "Betahistine" (tablets) njani? Imiyalelo yokusebenzisa, ncomo, iinkcazelo kunye neempawu ichiza zithiwe thaca apha ngasezantsi. Ukongeza, siza kukuxelela into sixhobo eyabelwe, ziyimalini iindleko, ukuba ngaba uneziphumo ebezingalindelekanga kunye Izimo.

Ekwakhiweni, inkcazo imilo kunye

uhlobo Ukukhutshwa beziyobisi kwenye - iipilisi. Noko ke, ukuba ziyafumaneka ezishiyanayo izixa ukwimo esebenzayo:

  • Valium amacwecwe ezimhlophe imilo setyhula enombhalo lidle esisebenza (betahistine dihydrochloride) - 8 mg.
  • tablet lume kunye biconvex kunye amathamo elintlangothi ajikelezayo oneelebhile esisebenza (betahistine dihydrochloride) - 16 okanye ezingama-24 mg.

Njengoko izithako abangabancedani iinkcukacha zemilo ziqulathe sodium lauryl sulfate, isodiyam croscarmellose, microcrystalline kwincindi, nemagnesium stearate kunye citric acid.

Isenzo amayeza ye ichiza

Yintoni na ichiza "Betahistine?" Imiyalelo zokusetyenziswa (ixabiso amayeza ezidweliswe ngezantsi) uchaza ukuba ichiza yi-analogu ye histamine, leyo wadalwa izithako.

macwecwe Active nto ekwaziyo zibandakanya histamine H-3 no H-1 receptors (strong kunye bachasene buthathaka) CNS (ngamanye amazwi, receptors ze eziba vestibular neendlebe angaphakathi).

Emva kokuba imithi kwangoko kuchaphazela ukuhamba kwegazi, ekukhuthazeni ukukhuthazwa microcirculation kunye permeability le emithanjeni indlebe engaphakathi. Kwakhona, icandelo esebenzayo le medicament akwazi ukuzinzisa uxinzelelo kwi njengecochlea endolymph.

Ngenxa yokuba "Betahistine" yi inhibitor ye H 3 receptors nuclei inkqubo vestibular, asinto ibe nafuthe ngokukhawuleza kwi CNS. Ngenxa yoko, ichiza ingqalelo omeleza ukosuleleka (neuronal) luvo kwi nucleus vestibular.

Njengoko ithamo ekunene amayeza, unako ngokukhawuleza ngokwaneleyo ukuze kupheliswe iimpawu vertigo vestibular. Ixesha ukungakhuseleki isithako esebenzayo beziyobisi ujongene imizuzu embalwa ukuba ngenye imini.

inani rhoqo ichiza phantsi kweliso likagqirha kunciphisa kwezenzo nesiyezi, kunciphisa iithowuni kunye unkenteza ezindlebeni, wobuya azimise ukuva kwi kubola kwayo.

Olu nyango akanalo umthomalalisi kwaye a wu endli yokuphazamiseka uququzelelo.

iipropati pharmacokinetic

Drug "Betagestin" ukusuka vertigo ako ngokukhawuleza nangokupheleleyo. Its lamanani igazi eliyincopho ziyaphunyezwa malunga nowama-65 imizuzu emva kokuthatha azila ukudla.

Iziyobisi elikhutheleyo medicament ezinxulumene neprothini ngaphantsi kwe-5%.

Isuselwe iziyobisi lokugaya ku metabolites engasebenziyo - demetilbetagistina no-2-pyridylacetic acid. Ukupheliswa phantse epheleleyo ichiza kwenzeka ngexesha lasemini ngokusebenzisa izintso (90%). Kuba i-10%, baya ziboniswa emathunjini.

Ubungqina obubonakalayo buxela

Drug "Betagestin" ukusuka nesiyezi eyabelwe izigulane rhoqo kakhulu. Ukongeza, iyeza ezisetyenziselwa ukunyanga Meniere engqondweni, kwakunye ukuphelisa ingxolo ezindlebeni, isicaphucaphu, ilahleko yokungeva kakuhle kunye nokulungelelaniswa kakuhle.

Kufuneka kuqatshelwe ukuba Meniere kaThixo syndrome ubonisa njengoko iingxaki izandi vestibular ukuba zange ngaphambili awayezibona ebantwini. Kwakhona kwenzeka ngohlobo kokubetha ahlekise. Meniere engqondweni na amathuba ophezulu likakade rhoqo.

Izimo

Ngoku uyazi iinjongo apho ichiza elisetyenziswa "Betagestin". Ukusuka vertigo ezigcinayo kakuhle kakhulu. Nangona kunjalo, eli chiza kukho Izimo. Kumele ukuba kumiselwe kubantu pheochromocytoma.

Ekubeni ichiza esebenzayo i analogu zokwenziwa of histamine, ukusetyenziswa kwayo ukuze negalelo nokukhululwa catecholamines, nto leyo ekhokelela wegazi kakhulu.

Kufuneka kuqatshelwe ukuba icebo lika "betahistine" Amacwecwe ukuba contraindicated kwizigulane kunye hypersensitivity yecandelo esebenzayo, okanye naziphi na ezinye excipients ngaphakathi nokwakheka ichiza.

imiyalelo iziyobisi

Drug "Betagestin" ukusuka vertigo kufuneka zithathwe ngqo ngokwemiyalelo enikwe.

  • Esithathwa kwizigulane abadala.

"Betahistine" macwecwe yayisalawulwa izilinganiso 8 okanye 16 mg kathathu ngemini (ekuqaleni konyango) kunye isidlo okanye emva kwayo. Ithamo yesondlo yahluka amayeza 24-48 mg ngosuku (ngokokubona kagqirha).

akufuneki ibe ngaphezulu kwama-48 mg idosi yemihla ngemihla ichiza. It lilungiswa zonke umguli ngamnye. Ngamanye amaxesha ukuphucula imeko yakhe ibonakala kuphela emva kweeveki ezimbalwa.

  • Unyango yabantu ngentliziyo, wezintso kwaye ukusilela wesibindi.

Izigulana ezo iSifo iziyobisi "Betahistine" uya kunyulwa kuphela emva kokuba axilongwe.

  • Unyango lwe abadala.

Ebudaleni ikwandim, ichiza kufuneka imiselwe ngokuqaphela okukhulu. Oku kungenxa yokuba kweli qela lwezigulane kukho amathuba okuba enkulu yeziphumo ebezingalindelekanga ezivela ephilayo izinto abangabancedani kwaye esebenzayo, eziyinxalenye amacwecwe.

  • Unyango abantwana abafikisayo.

Drug "Betagestin" ukusuka vertigo ungamiselwanga ukuba abantwana abafikisayo (neminyaka engaphantsi kwe 18). Oku kungenxa yokusilela ukusebenza kunye nokhuseleko amayeza data.

amacala libanda

Ukuba libanda, "Betahistine" ezithile izigulane zinokuba iimpawu ezifana isicaphucaphu, intloko ebuhlungu, iintlungu esiswini kunye ukozela (ngexesha uthatha ithamo ukuya ku-640 mg).

Kwakhona, izigulane ezikhala amahlaba, ukugabha, ukuqunjelwa, kunye Ataxia.

Ukuze iingxaki ezininzi kakhulu ziquka iingxaki sentliziyo miphungeni (yabonakala libanda ngabom).

Treatment - ukuhlamba esiswini kwisithuba semizuzu engama-60 emva kokuba yolawulo.

imiphumela emibi

Ayizizo zonke izigulane ezithatha ichiza "Betagestin", kungenzeka ubuhlungu.

Oogqirha ingxelo ukuba ngokubonakala reactions ezibi xa uthatha nawaphi na amayeza isigulane kunokuthetha zokuzama namayeza amatsha. Kule meko, qiniseka ukuba udibane nogqirha wakho phambi kokuba ukuphelisa ichiza.

ziphumo bezingalindelekanga Common ekuthatheni "betahistine" kuphawula omunye kwizigulana ezilishumi. Uluhlu iziphumo zixhaphakileyo ezibi ziquka iimpawu ezifana:

  • nesisu (ngokuqhelekileyo kwenzeka xa uthatha amayeza phambi kokuba isidlo);
  • umkhuhlane jikelele;
  • ubuhlungu okanye ukuqumba;
  • yintloko (ungathatha ntlungu, kodwa ke kuphela emva kokubonisana ngaphambi kunye specialist);
  • ziyabagulisa eluswini ngokohlobo sokudlathuka kweenwele krwada (kufuneka athathe iindawo ingxaki antihistamine okanye igrisi amafutha).

Ukuba izikhokelo akahambi kunceda ukuphelisa ziziphumo ebezingalindelekanga, isigulane kufuneka ubone ugqirha.

Ixabiso beziyobisi

Lwentengo "Betahistine" Amacwecwe inokuba nomahluko kwaye ixhomekeka kwisixa amayeza kwiphakheji. Amachiza ithamo of mg 24 zingathengwa ngenxa 60-65 engange. Izigulane ezininzi bakholelwa ukuba kakhulu sisiyobisi ixabiso eliphantsi.

Izimvo emithi

Izimvo "Betahistine" kuqulunqo ziyabethabethana. Ezinye izigulane abanezifo ezingapheliyo sentliziyo ukuthatha rhoqo amacwecwe. Noko ke, azisoloko ayisuse yintloko kunye nesiyezi.

Kunye nohlolo ngale medicament ezimbi nezilungileyo zibonisa ukuba ufuna isicelo okhethekileyo.

Ngoko, xa kakubi omnye ichiza "Betahistine" ungenza ngokukhawuleza ukubuyisela impilo kwisigulana, lo gama enye, phezu koko, akanaye yifuna, kodwa ukunciphisa kuphela imbonakalo iimpawu.

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