Zempilo, Ukulungiselela
"Flosteron": ukuhlaziywa. "I-Flosteron" yokunyamezela
Ngaba uyazi ukuba yintoni isilwanyana esinjenge "Flosteron"? Iingcali zithi le sixhobo esipheleleyo esingasetyenziselwa iintlobo ezahlukeneyo zesifo.
Ngokumalunga neliphi iipropati eli liliphi, liphi na uhlobo lokuthengwa kunye nendlela yokusebenzisa ngayo, siza kuxela kwinqaku elinikeziweyo.
Ukupakisha, ukubunjwa kunye nefomu yokukhululwa
Uphi i-"Flosteron" ithengiswa? Uphononongo lwabantu buchaza ukuba la mayeza angathengwa nayiphi na ikhemisi. Kwakhona, ezinye izigulane ziyalithumela nge-intanethi.
I-arhente iqukethe izithako ezisebenzayo ezifana ne-betamethasone disodium phosphate kunye ne-betamethasone dipropionate. Ukongezelela, ukubunjwa kwamachiza kubandakanya izinto ezincedisayo ngendlela ye-sodium chloride, i-sodium carmelose, i- polysorbate 80, i- sodium edetate, i-methylparaben, i- benzyl alcohol, i- hydrochloric acid, i-propylparaben, i-sodium hydrogenphosphate i-dihydrate, amanzi ahlambulukileyo kunye ne-polyethylene glycol.
Isilwanyana "u-Flosteron", esihlaziywa ngokuqhubekayo, sikhiqizwa njengokumiswa kweenjini. Itholakala kuma-ampoules (1 ml nganye) kwiiphakheji ezidibeneyo.
Pharmacodynamics
Usebenza njani unyango lwe "Flosteron"? Imiyalelo yokusetyenziswa (ukuphononongwa kweengcali kule sixhobo kuphela kuphela) iingxelo ukuba izinto ezichaphazelekayo zezidakamizwa ziyi-glucocorticosteroids (oko kukuthi, indawo yokufakelwa kwama-hormones adrenal). Zine-immunosuppressive, anti-rheumatic and anti-inflammatory properties.
I-Betamethasone ithinta i-homeostasis ye-glucose, i-metabolism yamandla kunye ne-hormone yondlo nge-adenohypophysis.
Kuza kube yimhla, umgaqo wesenzo se-glucocorticosteroids ayizange ifundwe kuze kube sekupheleni. Nangona kunjalo, kukho uluvo lokuba inkqubo yefuthe labo lwenziwa kwinqanaba leselula. Iingcali zikholelwa ukuba kwi-cytoplasm yeseli kukho iinkqubo ezi-2 ze-receptor, kwaye i-betamethasone ichaphazela ngqo ukuthatha inxaxheba kwi-receptors ekhethekileyo ye-GCS. Ngako oko, i-receptors ye-mineralocorticoid inegalelo kumgaqo we-sodium-potassium metabolism kunye nokulinganisela kwamanzi-electrolyte.
I-Corticosteroids zibizwa ngokuba yizinto ezinqunyuliswa ngamafutha. Ziyakwazi ukungena kalula kwiimbumba zeeseli kwisitye ekujoliswe kuyo.
Ngaloo ndlela, isenzo sonyango esilucinga ngalo sisekelwe kwiinkqubo ezithile ze-biochemical ezenzeka kwinqanaba le-molecular.
Pharmacokinetics
I-betamethasone dipropionate iyancipha ngokuthe ngcembe, nangona ibonelela ngokusisigxina. Ngokuxhomekeke kwindlela yokulawulwa kweziyobisi, inokuphumeza umphumo jikelele okanye wendawo.
Uxinzelelo oluphezulu lweziyobisi emva kokulawulwa kwe-intraarticular kugqitywa emva kwemizuzu engama-30. Kwi-plasma yegazi, isichengisi sibopha kwiiprotheni ngokukhawuleza. Ikwazi ukungena ngokukhawuleza kwimimandla ye-histohematological, kubandakanywa nomqobo we-placental.
I-metabolism yesilwanyana iqhutyelwa esibindi kunye nokubunjwa kweemetabolites ezingasebenzi. Ukuphuma kwezinto ezisebenzayo kwenzeka ngeentso, kunye kunye ne-bile kunye nentsasa yonina.
Iinkcazo
Xa izigulane zichazwe ijoyi ze "Flosteron"? Oogqirha bathi le yiyobisi yendalo yonke engasetyenziswa ekuphatheni izifo ezahlukahlukeneyo. Ngokwemiyalelo, eli gama lisetyenziswe xa:
- I-Edema yengqondo;
- Ukumpontshelwa igazi, ukukhathazeka, ukutshisa, i-anaphylactic, ugqirha, ukukhathazeka kwegazi kunye neentshutshiso ezinobuthi;
- Izifo zeethambo ezixhamlayo zendalo (ngokomzekelo, xa kwenzeka i-lupus erythematosus, ingxaki ye-thyrotoxic, i-coma ye-hepatic, i- rheumatoid arthritis);
- Unyango lwe-asthma ekhululekile;
- Ukuphendula kweAnaphylactoid ;
- Ukuthintela ukuvuvukala kunye nokukhawulwa emva kokubhenca kwi-cauterizing fluids.
Ndiyakwazi ukusebenzisa i-Flosteron ngenxa yokugula? Iingcali zithi le nkunkuma iphumelele kakhulu kwiimpendulo. Ngako oko, kudlalwa ukuba:
- I-asthma ye-Bronchial, i-rhinitis engapheliyo okanye yonyaka;
- I-Psoriasis, qhagamshelana ne-atopic dermatitis ne-keloid;
- Collagenoses;
- I-rheumatism eyongezelelweyo, i-lumbago, i-tendosynovitis, i-myositis, i-synovitis, i-post-traumatic osteoarthritis, i-epicondylitis, i-fibrositis;
- Ukulunywa kwezilwanyana;
- Zonke iintlobo zeempendulo ezithintekayo;
- Ulcerative colitis.
Ukungqinelana
Xa ungayisebenzisi nini le nkunkuma "Flosteron" (umyalelo, ukuphononongwa malunga nalo myeza kuza kuboniswa ngezantsi)? Akwabiwe xa:
- I-osteoporosis, isilonda esiswini, isifo sofuba, izifo ezithintekayo, i-glaucoma;
- Isenko-Cushing syndrome, thrombophlebitis, i-viral virus, i-fungal okanye i-bacterial infections, isifo sikashukela;
- Ukusebenza okukhulu kunye nokulimala, ngaphambi nangemva kokugonywa (kwiiveki ezimbini);
- I-Thrombocytopenic idiopathic purpura (intramuscular);
- Ukungabi nokuvuvukala kwamalungu;
- Ukuguqulwa kwamathambo kunye nokutshabalaliswa kokubambisana, ukungazinzi kokubambisana;
- Ukuphuma kwintsholongwane okanye ngenxa yokusetyenziswa kwama-antiticoagulants;
- Abesetyhini abasetyhini, abantwana abangaphantsi kweminyaka emithathu ubudala, i-hypersensitivity.
"I-Flosteron" amayeza: imiyalelo yokusetyenziswa
Izimvo zesigulane malunga nale nkunkuma zixube kakhulu.
Ndingayisebenzisa njani le chiza?
Ukuthatha umzimba kwisigulane somzimba, amayeza alawulwa nge-intramuscularly. Iilenki zenziwa kwi-gluteus muscle (inzulu) ngo-0.1-0.2 ml nganye kwiiveki ezi-2-4.
Uthi "u-Flosteron" unikwe njani ukunyamezela? Iingcali zithi eso sixhobo sisoloko sisetyenziselwa ukuvela kweempembelelo ezinobungozi. Kule meko, iilenki zenziwe nge-intramuscularly kwi-1-2 ml (kanye).
Ngokusetyenziswa kwesicatshulwa, i-dosage ingahluka kakhulu. Njengomthetho, ngu-0.25-2 ml.
I-psoriasis, i-neurodermatitis, i-eczema kunye nezinye izifo zesikhumba, amayeza alawulwa nge-intradermally.
Ukuba kuyimfuneko, le nkunkuma ingaxutywa kunye neprocaine okanye i-lidocaine ngenxa yokuphulukana nentlungu.
Kubantwana abaneminyaka engama-3-5, i-dose yokuqala yeli chiza i-0.3 ml, kunye nabantwana abama-6-12-0.6 ml.
Isiza "Flosteron": ukuhlaziywa
Ukuhlalutya iingcamango zeengcali malunga neziyobisi ngokubhekiselele kulo, zingagqiba ngokugqibeleleyo ukuba le nkunkuma iyasebenza kakhulu. Ngokutsho koogqirha, eli liyeza lisetyenziselwa izifo ezinzulu zeengqondo, izicubu ezixhamlayo, ukuphendula kwe-anaphylactoid, njl njl.
Ngokubhekisele kwizigulane, abahlala beshiya ingxelo emihle malunga nokumiswa kuka-Flosteron. Ubungqina bokuba abantu bathi le nyeza idla ngokuphindaphindiweyo. Ezi zibandakanya ukungcola, i-malaise jikelele, ukunqunyulwa kwesikhumba, ukufumana ubunzima nokunye okunjalo.
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