Zempilo, Amalungiselelo
"Tenorik": ncomo oogqirha. Amacwecwe ubunzima obungakumbi
Isebenza ukuba onjalo ichiza, njengoko "Tenorik"? Hlola eli chiza nga ushiye nganye. Ngokusebenzisa unxibelelwano ezinjalo kunye koogqirha kunye nezigulane kulula ukuba siphethe njani medicament wathi, nokuba ibangela reactions ecaleni kunye nokuba ukumelana msebenzi.
Kweli nqaku mayichaze ngokunzulu iimpawu kunye neempawu "Tenorik" iziyobisi. Hlola isigulane ukuthatha imiyalelo ugqirha wakhe, kuya kuba ngaphantsi kancinci nayo.
Ekwakhiweni, imilo, inkcazelo, ukupakishwa
Ukulungiselela "Tenorik" (100, 50 mg) liyahlonyelwa nawokwazisa ngawo amacwecwe emhlophe setyhula kunye imilo biconvex kunye mgca.
Ubume bale iyeza iqulethe izithako ezimbini ezisebenzayo: chlorthalidone kunye atenolol. Kwakhona, le kuqulunqo iqulathe amacandelo ezingaphezulu zinikiwe uhlobo lwengqolowa wesitatshi, isodiyam lauryl sulfate, lactose, polyvinylpyrrolidone, talc, dust, nemagnesium stearate kunye isopropanol.
Asinako ukuba ipilisi "Tenorik" (a uphengululo malunga esi sixhobo, ungabona ekupheleni kweli nqaku) zizele yayisoma bhanya okhethekileyo. Le ibandakanya methylene chloride, isopropanol, talc, hypromellose, titanium dioxide, macrogol neoli vaseline.
Zuza ingqalelo ichiza banokuba Imiqulu blister okanye imicu iipilisi 28 okanye 100.
Imithi Pharmaceutical Products
Yintoni iipilisi 'Tenorik "? Imiyalelo yokusebenzisa (iziyobisi ixabiso ayikho phezulu kakhulu) uchaza ukuba olu dibaniso arhente umfutho, onako ukwenza isiphumo iqinile ixesha elide.
Ukusebenza ichiza ethathelwa ingqalelo ngenxa isenzo ohlukileyo-2, okanye mandithi umchamo (chlorthalidone) kunye beta1-adrenergic blocker (atenolol).
iipropati key
atenolol ebizwa cardioselective beta1-blocker. Ukukwazi ukukhetha ngayo izinto lehla nge ukwandisa umthamo ichiza. Atenol akanayo inwebu yangaphakathi ekuzinziseni neziphumo sympathomimetic. Kanye njengezinye beta-blocker, iba nefuthe elibi inotropic kwaye ithintela kakhulu izinga intliziyo.
Yona chlorthalidone, kuyinto umchamo (sulfonamide netiazidny). It kwandisa ukhetho lweziqalelo ezifana chlorine kesodiyam. Kwakhona eli candelo kwandisa secretion of yesoda, magnesium potassium. Umgaqo wesenzo umfutho inxulunyaniswa sodium zinomgutyulo.
Atenolol kunye womchamo iphumelela kakhulu kunokuba ukusetyenziswa ngalinye kula ngokwahlukileyo.
Action ingqalelo ichiza kulo lonke ngosuku (emva idosi enye kwi idosi yemihla ngemihla).
Le kinetics beziyobisi
Ngenxa yokuba "Tenorik" analogs ichiza, ixabiso apho ziboniswa ngezantsi, yindlela zidibene siqwalasele iimpawu kwikinetiki nganye izinto esebenzayo ngokwahlukeneyo.
Atenolol ifunxwe yi 40-50% ukusuka phecana zesisu. eliphezulu Ayithandi ekufikelelwe kuso emva kweeyure-4 emva nokudla tablet. Unxibelelwano kunye neeproteni nama-8-16%.
Atenolol nto lakufumana yokucolwa wabonakalisa eqaqambileyo esibindini. Malunga ne-90% kwezi zinto wendele idubule ayitshintshanga iiyure 8-9. Eli xesha kufuneka zandiswe ukusilela kakhulu kwezintso, ukususela ukususwa atenolol lwenziwa yi nezintso.
Yona chlorthalidone, akukho 60% etsalwe iphecana zesisu. Xi plasma ifikelele iphezulu emva kweeyure ezili-12. Unxibelelwano kunye neeproteni ze nama-75%.
Chlorthalidone iboniswa yi izintso kwisithuba seeyure ezingama-50.
Ubungqina obubonakalayo buxela
Ukusuka ukunyuka koxinzelelo iziyobisi ingqalelo inceda kakuhle kakhulu. Eneneni, umfutho wegazi, yaye kuyinto enkulu, yaye mhlawumbi ebonisa kuphela ukusetyenziswa.
Izimo
Ngoku, uyazi, yintoni injongo linokukwenziwa "Tenorik" iipilisi (ezibonisa ukuba eli yeza zaye uchazwe apha ngasentla). Kodwa ke, ngelishwa, akukho ingqalelo ichiza kunye uluhlu khorwisaka Izimo. Ayikhuthazwa ukuthatha:
- yashiya cardiogenic;
- pheochromocytoma;
- bradycardia (wavakalisa uhlaselwe);
- izifo kakhulu ejikelezayo peripheral;
- hypotension (bedlulela esibi);
- lactic metabolic;
- AV-ukuvimba 1 nezinga 3;
- SSS;
- isifuba okuqhubekayo;
- senhliziyo (zombini etsolo kunye ezingapheliyo);
- diabetes;
- angina vasospastic (angina Prinzmetal yakhe);
- sifo;
- kwemigudu obstructive;
- hepatitis olunamandla;
- hypoglycemia;
- ukusilela kwezintso kwifomu oyingozi;
- ngaphantsi kweminyaka eli-18;
- myasthenia gravis;
- hypersensitivity ukuba izithako amayeza.
Indlela ukuthatha "Tenorik" high blood pressure?
izigulane abadala ezithatha ichiza kwixesha eliphakathi ekucetyiswa umthamo 100 mg. Ithamo yokuqala ichiza kufuneka mg 50 kanye ngemini.
Njengoko abantu abadala, ichiza "Tenorik" abelwe ukuba izixa kakhulu.
Izigulane nokusebenza kakuhle kwezintso Kuyancomeka ukunciphisa amaza ukuthatha iipilisi.
Kufuneka kuqatshelwe ukuba emva ukusetyenziswa elide ichiza uphononongwayo, ukurhoxiswa yayo iyafuneka ukuze afeze ngcembe.
imiphumela emibi
Reception "Tenorik" Amacwecwe ukuze bandiqumbise abasabela ecaleni zilandelayo:
- bradycardia, ukusilela ukwanda intliziyo, kwiziphelo ezibandayo, hypotension intolerance, arrhythmia, AV-block, iimpawu claudication ngakanye, Raynaud engqondweni ;
- ukudideka, silale, intloko ebuhlungu, ukuba nemibono, ukugula ngengqondo ebukhali, paresthesia, utshintsho kwimo, isiyezi, ukudinwa, sokulibala, nokudideka, ukungaboni;
- umlomo owomileyo, transaminases zesibindi kakhulu, ukuphazamiseka emathunjini, hepatotoxicity kunye cholestasis intrahepatic, pancreatitis, isicaphucaphu, ukuqhina, unesifo;
- leukopenia, purpura, thrombocytopenia, eosinophilia, agranulocytosis;
- alopecia, ukusabela psoriasiform, iliso owomileyo, exacerbation of ukhwekhwe, photosensitivity, isikhumba njengamaqhakuva;
- bronchospasm, hyperuricemia, hypokalemia, hyponatremia;
- kakuhle glucose ukunyamezelana, ukwanda kwenani omzimba antinuclear, kunciphise amandla.
Ezi ziphumo bezingalindelekanga zinqabile kunye nowobulali.
analogue Price
Amacwecwe Iindleko "Tenorik" ngu 110-120 engange. Bayakwazi indawo iziyobisi ezifana "Atenol", "Dinorik" okanye "Tenoret".
Izimvo amayeza "Tenorik"
Zokuvandlakanya impumelelo yale isixhobo selaybri ushiye nganye. Ngokutsho kwizigulane kunye amagqirha, okulungileyo esi sixhobo zezi:
- ukusebenza;
- ixabiso eliphantsi.
Bobubi kweli chiza ziquka:
- ukuba nokwenzeka ilahleko iinwele kunye nophuhliso yokungabi (ukhathalelo ixesha elide);
- amathuba okuvela ukuxhuzula.
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