Zempilo, Amalungiselelo
Efferalgan - imiyalelo yokusebenzisa
"Efferalgan" - a antipyretic ethandwayo. Nokubunjwa kwayo yahluke kancinane ngokuxhomekeke kwifom release. Ukubunjwa isiraphu abantwana - paracetamol kunye namacandelo abangabancedani: isiraphu, saccharin, polyethylene ethers, E202, izinongo, citric acid, amanzi okusela.
Standard iyafumaneka ezineengqayi iglasi kwi neelitha 0.09 (ngakumbi - icephe umlinganiselo).
Ukwakhiwa "Efferalgan" (efakwa): paracetamol, nezincedisi ezi semi-acylglycerol.
Umgangatho ngezi-amaqhosha-5, kwaye pack kukho 2 ukuphakheja.
Xa ukubunjwa effervescent iipilisi paracetamol kunye namacandelo abangabancedani: owomileyo isodium carbonate, povidone, citric acid, saccharin, sorbitol, isodiyam docusate, nesoda yokubhaka, E211.
La macwecwe amacwecwe-4, yonke impahla ye - kukho 4, uye iirekhodi 25.
imiphumela kwemithi
"Efferalgan" manual ichaza ichiza, iyeza engundoqo esebenzayo i paracetamol, apho iibhloko cyclooxygenase-1 no-2 ikakhulu kwi-CNS, ngaloo ndlela linegalelo kwi kumaziko thermoregulatory nentlungu. Zomzimba asha inyathelo paracetamol kwi Cox ezivaliweyo peroxidases ezizodwa, ezithile. Lo nto ichaza ukungabikho phantse ngokupheleleyo kwezinto anti-ukudumba esebenzayo. I-paracetamol ayikho nangayiphi na indlela kuchaphazele ukuyilwa prostaglandins zomzimba peripheral, nto leyo echaza ukungakwazi kwakhe okupheleleyo ukuphembelela isifo zesisu kunye nemali electrolyte-manzi.
Amakhandlela "Efferalgan" umyalelo libonisa zombini arhente ukuba iintlungu, isiphumo antiinflammatory kunye antipyretic engavezwanga.
I-paracetamol kudla ukudla ngokupheleleyo kwaye ngokukhawuleza. Le xi iphezulu kweziyobisi serum kwenzeka kwisithuba semizuzu 30-60. emveni kokuba besele. zasasazwa ngokukhawuleza kulo lonke ancedisana umzimba, paracetamol yakhiwe tenxileyo ubotshiwe kwiiproteni plasma (ukuya kwi-25%). Yena ingena umqobo segazi lobuchopho.
Sam nethe eveliswe sisibindi. I-paracetamol na Imveliso esuka emzimbeni metabolites. Oku kubonakaliswa luhlobo ephambili% 5 kuphela kuqulunqo.
ubungqina
Drug "Efferalgan" sikhokelo uncoma miqathango ilandelayo nezifo:
- zombini iziyobisi antipyretic phantsi eqhelekileyo OCR, ezimbi ebuntwaneni ezosulelayo, umkhuhlane, iingxaki postprivivochnyh, izifo ezosulelayo kunye kwiintetho ezikralayo, obubonakala ngokuba yincwadi evuliweyo komzimba;
- njengokuba iintlungu ngokulinganisela kwaye ezibuthathaka iintlungu (intloko ebuhlungu, iintlungu apha esihlunwini striated, iintlungu wamazinyo, izilonda luvo neuropathy, iintlungu, xa ukutsha, trauma).
Izimo
Izimo ekufumaneni "Efferalgan" umyalelo ibonisa onjalo (isibane, isiraphu)
- ezinkulu ukwaphulwa iinkqubo ze esibindini okanye yezintso;
- landa susceptibility yecandelo engundoqo;
- isifo igazi;
- ubudala kwinyanga enye (ukuba isiraphu) kwaye ukuya kwiinyanga ezintathu (ngokuba suppositories 0.08 g);
- abanalo enzyme G-6-PD;
- ukopha okanye iimpendulo ukudumba kwi isikali (suppository).
Ezithathwe ngononophelo ichiza kufuneka ube:
- ukuhluleka hepatic kwaye kwezintso (okt xa cholehemia usapho);
- in sezintso umsantsa ukusilela ubuncinane phakathi ukusetyenziswa yokulungiselela isiraphu - Iiyure ezi-8.
- hayi Kucetyiswa ukuba basebenzise amakhandlela urhudo.
Tablets "Efferalgan" umyalelo manual alukho kwi:
- anda susceptibility amacandelo;
- rhoqo (qho) ukusetyenziswa kotywala;
- Pregnancy (1 no-3 trimesters) kwaye ngethuba lokutyisa;
- abanalo enzyme G-6-PD;
- ngaphambi kokuba kubudala beminyaka elishumi elinesihlanu (ubunzima bomzimba - engaphantsi kwama-50 kg).
Tablets esithathwe isilumkiso:
- ukuphazamiseka kwesibindi kunye kidney umsebenzi;
- in senyongo naso (yeeFom ze-Johnson syndrome, cholehemia edluliselwa), hepatitis wentsholongwane egazini, ubudala ngaphezu 60 iilitha, isifo zesibindi (utywala) ..
imiphumela emibi
iziphumo ezingalindelekanga xa uthatha "Efferalgan" amagqabantshintshi zemiyalelo zezi:
- kunqabile kakhulu - ukugabha, isicaphucaphu, nokwaliwa (irhashalala, urticaria, pruritus, angioedema);
- umnqweno lobuxoki azikhulula futhi deurinatsii;
- ukudumba kwiinwebu isikali;
- kunqabile kakhulu - thrombocytopenia, igazi, igazi engaphezulu methemoglobin egazini ukuswela neutrophils leykotsitopeniya.
Ukuba unyango ixesha elide hi mpimo ngokugqithisileyo inokuba zinetyhefu kancinane kwesibindi kunye nezintso.
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