Zempilo, Amalungiselelo
"Dipyridamole": imiyalelo ukusetyenziswa. "Dipyridamole": imihlolo analogue
Yintoni na ichiza "Dipyridamole"? Imiyalelo, ixabiso, iimpawu, kunye ezibonisa ezi mali ziya thaca ngezantsi. Siya kunixelela ukuba kunokwenzeka ukufumana uthe iziyobisi ngexesha lokukhulelwa, ukuba wayenazo na analogue, iziphumo ebezingalindelekanga kunye Izimo.
Ubume, ukupakisha kunye nemilo
Ebonisa ukuba nolungiselelo yesikhokelo? "Dipyridamole" - ichiza ukuba unalo uhlobo ukukhululwa. Makhe siqwalasele ngokweenkcukacha ngaphezulu:
- Dragee 0.075 no 0.025, iyeza esebenzayo yale fomu dipyridamole. Ichiza kuthengiswa kupakisho zeplastiki lamaqhosha 100.
- "Dipyridamole" - amacwecwe 0,075, 0,005 no 0,025 g Camera, ukuba nayo ke into esebenzayo ezifana dipyridamole. Ngokuphathelele izinto abangabancedani, le yokugqibela ziquka icalcium stearate, monohydrate lactose nestatshi. Amayeza kuthengiswa blister iziqwenga 120 okanye ama-40, ezithi zibekwe imfumba kwikhadibhodi.
- A isisombululo ngenaliti. Le fom ubandakanya into esebenzayo efanayo. 0.5% isisombululo kuthengiswa nengqayi ye ml-2.
pharmacodynamics
Zeziphi iimpawu ingqalelo amayeza? Kuthetha ntoni apha imiyalelo ukusetyenziswa? "Dipyridamole" - ichiza ukuba unalo nomphumo vasodilating. Isenzo esinjalo it has ikakhulu nasezimpahleni ivaleke.
Umthamo owamkelweyo medicament abangaphangeliyo adhesion of zegazi kwandisa igazi isantya sokuqukuqela, iphucula kwaye iguqulela amanyathelo angioprotective. Ngaphezu koko, indlela isifundo ikhuthaza ukujikeleziswa collateral kwi iimpahla intliziyo.
Asinako ukuba ichiza normalizes ukuphuma lwemithambo. Ngoko ke, ukutya kwayo rhoqo kunciphisa kakhulu umngcipheko thrombosis, ingakumbi kwixesha postoperative.
isimiso ukusebenza
Yintoni enye chiza iipropati "Dipyridamole"? Manual ukuba kuthetha kakuhle lihlisa nethoni beempahla nedumbe lengqondo. Kule nkalo, Kuyinto ngokubonakalayo ukusetyenziselwa kukuhlaselwa idlule kobuchopho. Ngaphezu koko, oko ingqalelo ichiza kuphucula ejikeleza ephawulekayo placental. Olu phawu ikuvumela ukuba ukuthintela hypoxia Palsy.
Yintoni na indlela yesenzo ichiza? Yiyiphi inkcazelo iqulethe imiyalelo yokusebenzisa? "Dipyridamole" kwandisa umsebenzi adenosine kwaye kunciphisa kwizihlunu yayo okumbophelela. Yathi into kuchaphazela izihlunu nemithambo ngokubhloka release norepinephrine, leyo, enyanisweni, kubangele nokuncipha kwabo, uxinzelelo lwegazi kunye nokumelana systemic nemithambo.
Kwakhona kufanele kuqatshelwe ukuba ngenxa evalela i phosphodiesterase unciphisa kokukhutshwa activators udibaniso lwe ziiplatelets. Olu phawu likhusele unamathele. Ukwehla adhesiveness zegazi kuthintela egazi igazi nasemiphandeni.
Drug "Dipyridamole", ixabiso yayo eboniswe ngezantsi, njengoko arhente antiplatelet isoloko isetyenziswa ne acetylsalicylic acid.
Pharmacokinetics
Wendele ingqalelo indlela kunokuba ngokukhawuleza. eliphezulu Ayithandi ekufikelelwe kuso malunga nemizuzu engama-60 emva kokuba yolawulo.
Ukuqokelelela iziyobisi esebenzayo oluqhutywa myocardiocytes. Drug ivavanywa yokucolwa esibindini. Kwimeko zokugxojwa kulo mzimba yomsebenzi sokuzuza kunokwenzeka.
Ubungqina obubonakalayo buxela
Medicament "Dipyridamole" kumiselwe zifo zilandelayo:
- insufficiency coronary uhlobo ezingapheliyo;
- lokuthintela occlusion of shunts kunye stents;
- angina;
- iposi engabalulekanga (hayi kuphela kwisigaba oyingozi);
- lwemithambo kunye lwemithambo thrombosis;
- stroke kobuchopho;
- ukuthintelwa thromboembolism, ingakumbi emva kokuba ungenelelo zotyando entliziyweni;
- insufficiency placental;
- Encephalopathy yegazi;
- yamafutha imilenze;
- izifo microcirculatory nayiphi na imvelaphi;
- glomerulonephritis;
- DIC e nokudumba kwindawo umntwana toxicosis.
Izimo
Ngokutsho imiyalelo-mali ayikwazi ingasetyenziswa xa zokwahluka zilandelayo:
- hypotension ;
- angina eziguquguqukayo;
- iposi engabalulekanga olunamandla;
- hypersensitivity;
- arrhythmias kakhulu;
- senhliziyo decompensated;
- isibindi;
- sophele diathesis;
- isisu izilonda, ingakumbi eneengcinga ukopha.
Kufuneka kwakhona zithi le ichiza emiselweyo ngokuqaphela abantwana abangaphantsi kweminyaka eli-12 ubudala kunye zisanyisa. Ngaphezu koko, akunakwenzeka ukuba ukusebenzisa le arhente yegazi ngexesha yokuwa.
Imiyalelo yokusebenzisa
"Dipyridamole" - nechiza elichasene-thrombotic ekufuneka kuphela ngugqirha khona.
Ngokubanzi, amacwecwe kunye neepilisi athathwa ngomlomo imizuzu engama-60 ngaphambi kokuba kudliwe, iglasi yamanzi. Ukwenzela ukunciphisa isiphumo ukubacaphukisa kwi isifo esiswini ichiza nga mazihlanjwe phantsi ubisi efudumeleyo.
Umthamo kunye nendlela ukusetyenziswa ichiza kufuneka zifakelwe kuphela ngugqirha ngokuxhomekeke kubudala yesigulane, ukufunda kwakunye nemeko yempilo yakhe.
Kuthintelo thrombosis ezilawulwa 75 mg medicament amaxesha 6 ngosuku (idosi iphezulu yemihla ngemihla - 300-450 mg).
Xa insufficiency coronary usebenzisa 25-50 mg beziyobisi kathathu ngemini. Ithamo eliphezulu kule state - malunga 150-200 mg.
Ukuze kuthintelwe ekunqandeni le sihlume stent kwaye isigulane unikwa mg 50 ka iziyobisi (kane ngemini) kunye acetylsalicylic acid. Le medicament kusetyenziswa phambi kokuba ukusebenza, kwakunye nangexesha lokubhalwa ngeveki emva.
Xa izifo occlusive nemithambo ye nemilenze Kucetyiswa ukuba athathe 75 mg beziyobisi kathathu ngemini.
Idosi yemihla ngemihla ichiza ebantwaneni ixhomekeke ubunzima lwabo (5-10 mg ngalinye kg).
Ngokwemiyalelo, ngexesha unyango kuyimfuneko ukunciphisa ukuselwa iti nekofu, njengoko buthathaka isiphumo amayeza.
libanda
Xa usebenzisa ngeedosi eziphezulu beziyobisi mpawu zilandelayo kwenzeka isigulane: uxinzelelo lwegazi, isiyezi, ukunyuka kweqondo inhliziyo kwegazi. Kulo mzekelo, siyeke neziyobisi udibane nogqirha.
ukusabela ezingalunganga
Ngokutsho iimpendulo yezigulane, kwezinye iimeko, nangokwamkela imali kunokubangela iziphumo ebezingalindelekanga kulandelayo:
- ziyabagulisa;
- iyangongoza intliziyo;
- yandisa uxinzelelo lwegazi (ingakumbi xa zilawulwa yegazi);
- thrombocytopenia;
- intloko;
- izifo dyspeptic;
- ingxolo intloko;
- ukugungxula yobuso;
- tachycardia;
- ukopha ukwanda okanye ukopha.
imithi
ukusebenza Antiplatelet beziyobisi kunyuswa ulawulo ngaxeshanye kunye acetylsalicylic acid, tetracycline, penicillin, cephalosporin, anticoagulants ongangqalanga nicotinic acid.
Kufuneka kuqatshelwe ukuba anticoagulants ngqo, thrombolytics kunye lweeHedfowuni kungandisa okunokwenzeka yeengxaki ukopha.
Asikwazi ukuba amachiza caffeine kunye xanthine ukunciphisa vasodilating kunye neziphumo anti-thrombotic iimali ezo, kwaye asidi ukunciphisa ukufunxeka kwayo nokunciphisa ukufumaneka egazini.
Ngokumalunga kumalungiselelo kuchaziwe, kwenyusa imiphumo amachiza umfutho.
Ngaba ukusebenzisa amayeza "Dipyridamole" ngexa lokukhulelwa?
Iingcali zithi ngexesha uthatha phantsi imali ingqalelo abasetyhini abakhulelweyo ukuphuhlisa iingxaki. Ngokwahlukileyo koko, eli chiza "Dipyridamole" ngexesha lokukhulelwa udla emiselweyo xa kukho intsongelo kwesisu umntwana okanye insufficiency placental.
Amanani kunye analogue
Ichiza singavalwa "Dipyridamole"? Analogs-mali zidweliswe ngezantsi. Ezi zibandakanya ezi machiza alandelayo: "Parsedil", "Kurantil", "Padikor", "Antistenokardin", "Trankokord", "angina", "persantin", "Dipyridamole-Verein". Zonke ezi imithi eyona nto efanayo esebenzayo. Noko ke, ukuze abe neziphumo ebezingalindelekanga ezahlukeneyo Izimo. Kule meko, kucetyiswa ukuba usebenzise ezi mali kuphela emva kokudibana nogqirha wakho.
Yimalini sisiyobisi "Dipyridamole"? ixabiso layo isusela evela engange 380-420 (ngokuxhomekeke kwisixa kunye nefomu wokukhulula iziyobisi).
reviews
Amaninzi, impendulo yakho malunga nale sixhobo usele kwezo izigulane kuba lowo ukuba ezimiselweyo nokuthintela kunye nokunyanga yokuya ukuguga placental, kwakunye insufficiency placental.
Kufuneka kuqatshelwe ukuba abasetyhini abakhulelweyo ubunzima isiyobisi enjalo kuhle. Kuphela nje ezimbalwa besini enobulungisa ukuba basabele egwenxa ngohlobo ukwehliswa uxinzelelo lwegazi kunye nesiyezi.
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