Zempilo, Amalungiselelo
Drug "Tramal": ncomo, imiyalelo, izalathiso
analgesics opioid ebizwa arhente zokubambela kundlunkulu asetyenziswa womelele iintlungu syndrome. La machiza kufuneka nempembelelo ethile kwinkqubo luvo.
Kukho iziyobisi abaninzi propati. Enye yazo i "Tramal". Imiyalelo yokusebenzisa, ncomo, iimpawu, imbonakaliso kunye neziphumo ebezingalindelekanga ichiza zithiwe thaca apha ngasezantsi.
Form, ukwakheka
Le medicament "Tramal" ratings nto leyo ushiye ngamnye abe ezininzi iintlobo wokwenziwa: kuwisa yolawulo ngomlomo, njengezingxobo, suppositories, efakwa kunye inaliti. Eyona nto elikhutheleyo ichiza tramadol hydrochloride. Kwakhona amachiza ziquka izinto abancedisayo (kuxhomekeka kuhlobo lwe medicament).
iipropati kwemithi
Yintoni na ichiza "Tramal"? Ukuphonononga baxele ukuba iintlungu opioid. Anakho iipropati eyomeleleyo iintlungu, nto leyo wachaza neziphumo zayo agonist receptors elise CNS.
Le medicament yi opioid (zokwenziwa). It is a racemate of isomers ezimbi nezilungileyo izinto ngenye indlela inxaxheba kwisenzo iintlungu.
isomer Positive - yinto receptor opioid olunyulu agonist. Ngokuphathelele izinto ezingakhiyo, ngoko ke unako ukuze kuthintelwe kuhluthwe (neuronal) norepinephrine, kwakunye yenza esihla inkqubo central noradrenergic. Oku kukhokelela ukuphazamiseka ukosuleleka neemvakalelo intlungu iziyobisi (gelatin) umnqonqo.
Zombini isomers zimelwe yi ngendlela ihambelana.
iziyobisi kujongwa ebangela umthomalalisi. Ngeedosi zonyango ngokoqobo loo nto ayithethi zinqanda ukusebenza kwenkqubo bokuphefumla alunasiphumo kwi hemodynamics.
Xa kulawulwa reception likhoboka neziyobisi kunye nokuxhomekeka ukuphuhlisa kunqabile. Ngendlela, xa ukusetyenziswa icaffeine na ucaca ngakumbi.
kinetics
ingaba ichiza wendele yi "Tramal"? Ukuphonononga baxele ukuba xa kuthatyathwa ngomlomo oko ifunxwe yi-90%.
Emva kokuba ulawulo intramuscular xi incopho beziyobisi egazini kwenzeka emva kweyure enye.
medicament kujongwa ingena umqobo placental kunye BBB. Yena umi kwakhona phandle ubisi lukanina.
Ukurhoxiswa ichiza ngokusebenzisa nezintso.
ubungqina
Kwezinye iimeko, iyeza efunekayo "Tramal"? Uphengululo (in Oncology le ukulungiselela isetyenziswa rhoqo kakhulu) lithi lithathwa kuthetha eboniswe syndrome intlungu ngobunzulu eyomeleleyo avareji imvelaphi ezahlukeneyo:
- ukuphatheka;
- ngexesha postoperative;
- ngokuba ntlungu kwenzeka ngenxa iposi engabalulekanga;
- buhlungu xa zisebenzisa iindlela zonyango okanye zokuxilonga.
Izimo
Xa kufuneka usebenzise amayeza "Tramal"? iingcali Guest lubonisa Izimo, ezifana:
- ukusetyenziswa esihamba ngayo inhibitors monoamine oxidase, kwakunye iiveki ezimbini emva kokuba zokurhoxa zabo;
- iimeko zihambisana inhibition uphawu lwe CNS okanye ukudandatheka yokuphefumla (umz, Ityhefu utywala, analgesics opioid, psychotropic okanye iziyobisi thile kuthetha);
- ukusilela kwezintso, elibaleka yayinzima;
- ekubalekeni syndrome yemithi;
- ukusilela hepatic yayinzima;
- hypersensitivity.
Zonke ezi zinto kufuneka ithathelwe ingqalelo.
Drug "Tramal": imiyalelo yokusebenzisa
Lwezitofu, kwakhona kuya thaca ngezantsi, linokukwenziwa ukuba butofelwe, kwesikhumba okanye intramuscularly.
Ngaphakathi kule amayeza kufuneka amakathathwe phambi, ngexesha okanye emva kwesidlo. philisi yesiqhelo kwehle ngamanzi, kwaye nesisombululo ithe yawa phezu iqhekeza yeswekile okanye exutywe umthamo omncinci ulwelo.
Ke ukuba suppository efakwa ilawulwa kwi isikali.
Esithathwa beziyobisi ethathelwa ingqalelo xa kumiselwa kuxhomekeke kubungakanani intlungu.
Kwezinye iimeko, yenza izitofu 'Tramal "? Ukuphonononga zibonisa ukuba olu hlobo beziyobisi kusetyenziswa kuphela kwimeko ukuba ufuna ukufikelela isiphumo ngokukhawuleza iintlungu.
imiphumela emibi
Njengoko nabanye analgesics, ingqalelo ichiza kungabangela iintlobo ngayo kwicala ezifana:
- anozizi eluswini, isicaphucaphu, ukuxhuzula ebuchotsheni, umlomo owomileyo, ukudinwa, ukugabha;
- isiyezi, iintlungu esiswini, mgaqweni intliziyo isingqisho, esiswini;
- kutshintsha ukutya, ukozela, intloko ebuhlungu, tachycardia, utshintsho isimo, ukudakumba, abasabela kakuhle zokuziphatha, utshintsho kumsebenzi, ubunzima ukuginya emanzini;
- niphele, buthathaka kwezihlunu, ukuyisonga;
- irhashalala eluswini, ukuqhina, ubuthathaka iimoto, ukudideka, ukubila.
izincomo ezithile
Ngononophelo olukhulu ichiza emiselweyo ukuba abantu kumsebenzi othile wesibindi nezintso ngamandla ophakamileyo intracranial, iintlungu esiswini, ukwenzakala ebuchotsheni esibuhlungu, izigulane sokuwa, kwakunye ukuphazamiseka kwenkqubo sokuphefumla.
Ukusela utywala ngexesha unyango le arhente kumele isuswe.
reviews
izigulane ezininzi zithi ichiza "Tramal" i iintlungu esiqinileyo nesinempumelelo opioid. Naluphi na uhlobo nto intle ngokukhawuleza kususa nkqu syndromes kakhulu intlungu, lula kakhulu imeko yesigulane.
Bobubi olu nyango ziquka inani elikhulu reactions ezibi, kwakunye uluhlu khorwisaka Izimo.
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